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Structure-Guided Design of Substituted Biphenyl Butanoic Acid Derivatives as Neprilysin Inhibitors.
Kawanami, Toshio; Karki, Rajeshri G; Cody, Emma; Liu, Qian; Liang, Guiqing; Ksander, Gary M; Rigel, Dean F; Schiering, Nikolaus; Gong, Yongjin; Coppola, Gary M; Iwaki, Yuki; Sun, Robert; Neubert, Alan; Fan, Li; Ingles, Sara; D'Arcy, Allan; Villard, Frederic; Ramage, Paul; Jeng, Arco Y; Leung-Chu, Jennifer; Liu, Jing; Beil, Michael; Fu, Fumin; Chen, Wei; Cumin, Frederic; Wiesmann, Christian; Mogi, Muneto.
Affiliation
  • Kawanami T; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Karki RG; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Cody E; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Liu Q; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Liang G; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Ksander GM; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Rigel DF; Novartis Pharmaceuticals Corporation, One Health Plaza, East Hanover, New Jersey 07936-1080, United States.
  • Schiering N; Novartis Institutes for BioMedical Research, Novartis Campus, CH-4056 Basel, Switzerland.
  • Gong Y; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Coppola GM; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Iwaki Y; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Sun R; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Neubert A; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Fan L; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
  • Ingles S; Novartis Institutes for BioMedical Research, Novartis Campus, CH-4056 Basel, Switzerland.
  • D'Arcy A; Novartis Institutes for BioMedical Research, Novartis Campus, CH-4056 Basel, Switzerland.
  • Villard F; Novartis Institutes for BioMedical Research, Novartis Campus, CH-4056 Basel, Switzerland.
  • Ramage P; Novartis Institutes for BioMedical Research, Novartis Campus, CH-4056 Basel, Switzerland.
  • Jeng AY; Novartis Pharmaceuticals Corporation, One Health Plaza, East Hanover, New Jersey 07936-1080, United States.
  • Leung-Chu J; Novartis Pharmaceuticals Corporation, One Health Plaza, East Hanover, New Jersey 07936-1080, United States.
  • Liu J; Novartis Pharmaceuticals Corporation, One Health Plaza, East Hanover, New Jersey 07936-1080, United States.
  • Beil M; Novartis Pharmaceuticals Corporation, One Health Plaza, East Hanover, New Jersey 07936-1080, United States.
  • Fu F; Novartis Pharmaceuticals Corporation, One Health Plaza, East Hanover, New Jersey 07936-1080, United States.
  • Chen W; Novartis Pharmaceuticals Corporation, One Health Plaza, East Hanover, New Jersey 07936-1080, United States.
  • Cumin F; Novartis Institutes for BioMedical Research, Novartis Campus, CH-4056 Basel, Switzerland.
  • Wiesmann C; Novartis Institutes for BioMedical Research, Novartis Campus, CH-4056 Basel, Switzerland.
  • Mogi M; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts 02139, United States.
ACS Med Chem Lett ; 11(2): 188-194, 2020 Feb 13.
Article in En | MEDLINE | ID: mdl-32071687

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2020 Type: Article Affiliation country: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2020 Type: Article Affiliation country: United States