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Fragment-based discovery of orphan nuclear receptor Nur77/NGFI-B ligands.
Arifi, Silvia; Zaienne, Daniel; Heering, Jan; Wein, Thomas; Zhubi, Rezart; Chaikuad, Apirat; Knapp, Stefan; Marschner, Julian A; Merk, Daniel.
Affiliation
  • Arifi S; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Zaienne D; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Heering J; Fraunhofer Institute for Translational Medicine and Pharmacology ITMP, 60596 Frankfurt, Germany.
  • Wein T; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Zhubi R; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany; Structural Genomics Consortium, BMLS, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Chaikuad A; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany; Structural Genomics Consortium, BMLS, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Knapp S; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany; Structural Genomics Consortium, BMLS, Goethe University Frankfurt, 60438 Frankfurt, Germany.
  • Marschner JA; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany.
  • Merk D; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany; Department of Pharmacy, Ludwig-Maximilians-Universität München, 81377 Munich, Germany. Electronic address: daniel.merk@cup.lmu.de.
Bioorg Chem ; 129: 106164, 2022 12.
Article in En | MEDLINE | ID: mdl-36162288

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Receptors, Steroid / Neoplasms Type of study: Prognostic_studies Limits: Humans Language: En Journal: Bioorg Chem Year: 2022 Type: Article Affiliation country: Germany

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Receptors, Steroid / Neoplasms Type of study: Prognostic_studies Limits: Humans Language: En Journal: Bioorg Chem Year: 2022 Type: Article Affiliation country: Germany