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Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core.
Tîntas, Mihaela-Liliana; Peauger, Ludovic; Alix, Florent; Papamicaël, Cyril; Besson, Thierry; Sopková-de Oliveira Santos, Jana; Gembus, Vincent; Levacher, Vincent.
Affiliation
  • Tîntas ML; INSA Rouen Normandie, Univ. Rouen Normandie, CNRS UMR 6014 COBRA, FR 3038, F-76000 Rouen, France.
  • Peauger L; VFP Therapies, 15 rue François Couperin, 76000 Rouen, France.
  • Alix F; VFP Therapies, 15 rue François Couperin, 76000 Rouen, France.
  • Papamicaël C; INSA Rouen Normandie, Univ. Rouen Normandie, CNRS UMR 6014 COBRA, FR 3038, F-76000 Rouen, France.
  • Besson T; INSA Rouen Normandie, Univ. Rouen Normandie, CNRS UMR 6014 COBRA, FR 3038, F-76000 Rouen, France.
  • Sopková-de Oliveira Santos J; UNICAEN, CERMN (Centre d'Etudes et de Recherche sur le Médicament de Normandie), Normandie Univ., Bd Becquerel, F-14032 Caen, France.
  • Gembus V; VFP Therapies, 15 rue François Couperin, 76000 Rouen, France.
  • Levacher V; INSA Rouen Normandie, Univ. Rouen Normandie, CNRS UMR 6014 COBRA, FR 3038, F-76000 Rouen, France.
Molecules ; 28(1)2022 Dec 21.
Article in En | MEDLINE | ID: mdl-36615235

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinones / Protein Kinase Inhibitors Limits: Humans Language: En Journal: Molecules Journal subject: BIOLOGIA Year: 2022 Type: Article Affiliation country: France

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinones / Protein Kinase Inhibitors Limits: Humans Language: En Journal: Molecules Journal subject: BIOLOGIA Year: 2022 Type: Article Affiliation country: France