Your browser doesn't support javascript.
loading
First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53.
Nowak, Radoslaw P; Tumber, Anthony; Hendrix, Eline; Ansari, Mohammad Salik Zeya; Sabatino, Manuela; Antonini, Lorenzo; Andrijes, Regina; Salah, Eidarus; Mautone, Nicola; Pellegrini, Francesca Romana; Simelis, Klemensas; Kawamura, Akane; Johansson, Catrine; Passeri, Daniela; Pellicciari, Roberto; Ciogli, Alessia; Del Bufalo, Donatella; Ragno, Rino; Coleman, Mathew L; Trisciuoglio, Daniela; Mai, Antonello; Oppermann, Udo; Schofield, Christopher J; Rotili, Dante.
Afiliación
  • Nowak RP; Botnar Research Centre, Nuffield Orthopaedic Centre, University of Oxford, Headington OX3 7LD, U.K.
  • Tumber A; Botnar Research Centre, Nuffield Orthopaedic Centre, University of Oxford, Headington OX3 7LD, U.K.
  • Hendrix E; Chemistry Research Laboratory, Department of Chemistry and the Ineos Oxford Institute for Antimicrobial Research, 12, Mansfield Road, University of Oxford, Oxford OX1 3TA, U.K.
  • Ansari MSZ; Institute of Cancer and Genomic Sciences, University of Birmingham, Edgbaston, Birmingham B15 2TT, U.K.
  • Sabatino M; Institute of Molecular Biology and Pathology (IMBP), National Research Council (CNR) c/o Department of Biology and Biotechnology "Charles Darwin" Sapienza University of Rome, Via degli Apuli 4, Rome 00185, Italy.
  • Antonini L; Rome Center for Molecular Design, Department of Chemistry and Technology of Drugs, ″Sapienza″ University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy.
  • Andrijes R; Rome Center for Molecular Design, Department of Chemistry and Technology of Drugs, ″Sapienza″ University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy.
  • Salah E; Institute of Cancer and Genomic Sciences, University of Birmingham, Edgbaston, Birmingham B15 2TT, U.K.
  • Mautone N; Chemistry Research Laboratory, Department of Chemistry and the Ineos Oxford Institute for Antimicrobial Research, 12, Mansfield Road, University of Oxford, Oxford OX1 3TA, U.K.
  • Pellegrini FR; Department of Chemistry and Technology of Drugs, ″Sapienza″ University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy.
  • Simelis K; Institute of Molecular Biology and Pathology (IMBP), National Research Council (CNR) c/o Department of Biology and Biotechnology "Charles Darwin" Sapienza University of Rome, Via degli Apuli 4, Rome 00185, Italy.
  • Kawamura A; Chemistry Research Laboratory, Department of Chemistry and the Ineos Oxford Institute for Antimicrobial Research, 12, Mansfield Road, University of Oxford, Oxford OX1 3TA, U.K.
  • Johansson C; Chemistry - School of Natural and Environmental Sciences, Newcastle University, Newcastle upon Tyne NE1 7RU, U.K.
  • Passeri D; Botnar Research Centre, Nuffield Orthopaedic Centre, University of Oxford, Headington OX3 7LD, U.K.
  • Pellicciari R; Chemistry Research Laboratory, Department of Chemistry and the Ineos Oxford Institute for Antimicrobial Research, 12, Mansfield Road, University of Oxford, Oxford OX1 3TA, U.K.
  • Ciogli A; TES Pharma S.r.l. Via P. Togliatti 20, Corciano, Perugia 06073, Italy.
  • Del Bufalo D; TES Pharma S.r.l. Via P. Togliatti 20, Corciano, Perugia 06073, Italy.
  • Ragno R; Department of Chemistry and Technology of Drugs, ″Sapienza″ University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy.
  • Coleman ML; Preclinical Models and New Therapeutic Agents Unit, IRCCS-Regina Elena National Cancer Institute, Via Elio Chianesi 53, Rome 00144, Italy.
  • Trisciuoglio D; Rome Center for Molecular Design, Department of Chemistry and Technology of Drugs, ″Sapienza″ University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy.
  • Mai A; Institute of Cancer and Genomic Sciences, University of Birmingham, Edgbaston, Birmingham B15 2TT, U.K.
  • Oppermann U; Institute of Molecular Biology and Pathology (IMBP), National Research Council (CNR) c/o Department of Biology and Biotechnology "Charles Darwin" Sapienza University of Rome, Via degli Apuli 4, Rome 00185, Italy.
  • Schofield CJ; Department of Chemistry and Technology of Drugs, ″Sapienza″ University of Rome, Piazzale Aldo Moro 5, Rome 00185, Italy.
  • Rotili D; Botnar Research Centre, Nuffield Orthopaedic Centre, University of Oxford, Headington OX3 7LD, U.K.
J Med Chem ; 64(23): 17031-17050, 2021 12 09.
Article en En | MEDLINE | ID: mdl-34843649
Asunto(s)
Texto completo
Imprimir
XML
PubMed Links
Buscar en Google

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Ribosomas / Proteínas Nucleares / Dioxigenasas / Inhibidores Enzimáticos / Histona Demetilasas Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2021 Tipo del documento: Article País de afiliación: Reino Unido
Texto completo
Imprimir
XML
PubMed Links
Buscar en Google

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Ribosomas / Proteínas Nucleares / Dioxigenasas / Inhibidores Enzimáticos / Histona Demetilasas Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2021 Tipo del documento: Article País de afiliación: Reino Unido