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Structure optimization and discovery of novel compound for the treatment of insertion mutations within exon 20 of EGFR and HER2.
Cui, Yetong; Wang, Ruonan; Wei, Yujiao; Hou, Fei; Li, Haixi; Jiang, Yurui; Sun, Yue; Fu, Shushu; Zuo, Lina; Wang, Xiaoji; Li, Ming; Li, Jinling; Liu, Ning; Zhang, Kun; Wei, Mingming; Yang, Guang.
Afiliación
  • Cui Y; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China.
  • Wang R; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China.
  • Wei Y; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China.
  • Hou F; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China.
  • Li H; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China.
  • Jiang Y; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China.
  • Sun Y; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China.
  • Fu S; Engineering Research Center of Health Food Design & Nutrition Regulation, School of Chemical Engineering and Energy Technology, Dongguan University of Technology, Dongguan, 523808 Guangdong Province, PR China.
  • Zuo L; Engineering Research Center of Health Food Design & Nutrition Regulation, School of Chemical Engineering and Energy Technology, Dongguan University of Technology, Dongguan, 523808 Guangdong Province, PR China.
  • Wang X; Engineering Research Center of Health Food Design & Nutrition Regulation, School of Chemical Engineering and Energy Technology, Dongguan University of Technology, Dongguan, 523808 Guangdong Province, PR China. Electronic address: wangxj@dgut.edu.cn.
  • Li M; Cangzhou Institutes for Food and Drug Control, Cangzhou, 061000 Hebei Province, PR China. Electronic address: 83991223@qq.com.
  • Li J; Kangtai Pharmceutical Co. Ltd of Hebei, Cangzhou, 061000 Hebei Province, PR China. Electronic address: jinoplk@qq.com.
  • Liu N; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China. Electronic address: liuning@nankai.edu.cn.
  • Zhang K; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China. Electronic address: zhangkun1112@163.com.
  • Wei M; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China. Electronic address: mingmingshengwu@163.com.
  • Yang G; The State Key Laboratory of Medicinal Chemical Biology, College of Pharmacy, Nankai University, Tianjin 300071, PR China. Electronic address: guang.yang@nankai.edu.cn.
Bioorg Med Chem ; 81: 117202, 2023 03 01.
Article en En | MEDLINE | ID: mdl-36804726

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Carcinoma de Pulmón de Células no Pequeñas / Neoplasias Pulmonares Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Carcinoma de Pulmón de Células no Pequeñas / Neoplasias Pulmonares Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article