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Identification of potential inhibitors of casein kinase 2 alpha of Plasmodium falciparum with potent in vitro activity.
Tomaz, Kaira C P; Tavella, Tatyana A; Borba, Joyce V B; Salazar-Alvarez, Luis C; Levandoski, João E; Mottin, Melina; Sousa, Bruna K P; Moreira-Filho, José T; Almeida, Vitor M; Clementino, Leandro C; Bourgard, Catarina; Massirer, Katlin B; Couñago, Rafael M; Andrade, Carolina H; Sunnerhagen, Per; Bilsland, Elizabeth; Cassiano, Gustavo C; Costa, Fabio T M.
Afiliación
  • Tomaz KCP; Laboratory of Tropical Diseases (LDT), Institute of Biology, University of Campinas , Campinas, Brazil.
  • Tavella TA; Laboratory of Tropical Diseases (LDT), Institute of Biology, University of Campinas , Campinas, Brazil.
  • Borba JVB; Laboratory of Tropical Diseases (LDT), Institute of Biology, University of Campinas , Campinas, Brazil.
  • Salazar-Alvarez LC; Laboratory of Molecular Modeling and Drug Design (LabMol), Faculty of Pharmacy, Universidade Federal de Goiás (UFG) , Goiânia, Brazil.
  • Levandoski JE; Laboratory of Tropical Diseases (LDT), Institute of Biology, University of Campinas , Campinas, Brazil.
  • Mottin M; Department of Materials and Bioprocesses Engineering, School of Chemical Engineering, University of Campinas , Campinas, Brazil.
  • Sousa BKP; Laboratory of Molecular Modeling and Drug Design (LabMol), Faculty of Pharmacy, Universidade Federal de Goiás (UFG) , Goiânia, Brazil.
  • Moreira-Filho JT; Laboratory of Molecular Modeling and Drug Design (LabMol), Faculty of Pharmacy, Universidade Federal de Goiás (UFG) , Goiânia, Brazil.
  • Almeida VM; Laboratory of Molecular Modeling and Drug Design (LabMol), Faculty of Pharmacy, Universidade Federal de Goiás (UFG) , Goiânia, Brazil.
  • Clementino LC; Centro de Química Medicinal (CQMED), Centro de Biologia Molecular e Engenharia Genética(CBMEG), Universidade Estadual de Campinas (UNICAMP) , Campinas, Brazil.
  • Bourgard C; Laboratory of Tropical Diseases (LDT), Institute of Biology, University of Campinas , Campinas, Brazil.
  • Massirer KB; Laboratory of Tropical Diseases (LDT), Institute of Biology, University of Campinas , Campinas, Brazil.
  • Couñago RM; Department of Chemistry and Molecular Biology, University of Gothenburg , Gothenburg, Sweden.
  • Andrade CH; Centro de Química Medicinal (CQMED), Centro de Biologia Molecular e Engenharia Genética(CBMEG), Universidade Estadual de Campinas (UNICAMP) , Campinas, Brazil.
  • Sunnerhagen P; Centro de Química Medicinal (CQMED), Centro de Biologia Molecular e Engenharia Genética(CBMEG), Universidade Estadual de Campinas (UNICAMP) , Campinas, Brazil.
  • Bilsland E; Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill , Chapel Hill, North Carolina, USA.
  • Cassiano GC; Laboratory of Molecular Modeling and Drug Design (LabMol), Faculty of Pharmacy, Universidade Federal de Goiás (UFG) , Goiânia, Brazil.
  • Costa FTM; Center for Research and Advancement of Fragments and Molecular Targets (CRAFT), University of São Paulo , São Paulo, Brazil.
Antimicrob Agents Chemother ; 67(11): e0058923, 2023 11 15.
Article en En | MEDLINE | ID: mdl-37819090

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Plasmodium / Malaria Falciparum / Malaria / Antimaláricos Tipo de estudio: Diagnostic_studies / Prognostic_studies Idioma: En Revista: Antimicrob Agents Chemother Año: 2023 Tipo del documento: Article País de afiliación: Brasil

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Plasmodium / Malaria Falciparum / Malaria / Antimaláricos Tipo de estudio: Diagnostic_studies / Prognostic_studies Idioma: En Revista: Antimicrob Agents Chemother Año: 2023 Tipo del documento: Article País de afiliación: Brasil