RESUMEN
ACH-702 is a new isothiazoloquinolone with potent in vitro and in vivo activities against important bacterial pathogens, including Staphylococcus aureus. In this study, ACH-702 was found to have promising in vitro antibacterial activity against Mycobacterium tuberculosis, with MICs of Asunto(s)
Antituberculosos/farmacología
, Farmacorresistencia Bacteriana
, Mycobacterium tuberculosis/efectos de los fármacos
, Quinolonas/farmacología
, Tiazoles/farmacología
, Antituberculosos/química
, Girasa de ADN/genética
, Girasa de ADN/metabolismo
, Humanos
, Pruebas de Sensibilidad Microbiana
, Mycobacterium tuberculosis/aislamiento & purificación
, Quinolonas/química
, Tiazoles/química
, Inhibidores de Topoisomerasa II
, Tuberculosis/microbiología