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1.
Nonbisphosphonate inhibitors of Plasmodium falciparum FPPS/GGPPS.
Bioorg Med Chem Lett
; 41: 127978, 2021 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33766764
2.
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibition.
Bioorg Med Chem
; 24(11): 2486-503, 2016 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27112449
3.
Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel non-basic 1-(2H-indazole-5-yl)pyridin-2(1H)-one derivatives and mitigation of mutagenicity in Ames test.
Bioorg Med Chem
; 24(11): 2504-18, 2016 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27117261
4.
Design, Synthesis, and Evaluation of [18F]T-914 as a Novel Positron-Emission Tomography Tracer for Lysine-Specific Demethylase 1.
J Med Chem
; 64(17): 12680-12690, 2021 09 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-34423983
5.
Design and Synthesis of Novel Spiro Derivatives as Potent and Reversible Monoacylglycerol Lipase (MAGL) Inhibitors: Bioisosteric Transformation from 3-Oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl Moiety.
J Med Chem
; 64(15): 11014-11044, 2021 08 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-34328319
6.
Design and Identification of a GPR40 Full Agonist (SCO-267) Possessing a 2-Carbamoylphenyl Piperidine Moiety.
J Med Chem
; 63(18): 10352-10379, 2020 09 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-32900194
7.
Development of human cGAS-specific small-molecule inhibitors for repression of dsDNA-triggered interferon expression.
Nat Commun
; 10(1): 2261, 2019 05 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-31113940
8.
Design, Synthesis, and Evaluation of Piperazinyl Pyrrolidin-2-ones as a Novel Series of Reversible Monoacylglycerol Lipase Inhibitors.
J Med Chem
; 61(20): 9205-9217, 2018 10 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-30251836
9.
Publisher Correction: Small molecule inhibition of cGAS reduces interferon expression in primary macrophages from autoimmune mice.
Nat Commun
; 8(1): 1827, 2017 11 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-29170402
10.
Small molecule inhibition of cGAS reduces interferon expression in primary macrophages from autoimmune mice.
Nat Commun
; 8(1): 750, 2017 09 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-28963528
11.
Melanin-Concentrating Hormone Receptor 1 Antagonists Lacking an Aliphatic Amine: Synthesis and Structure-Activity Relationships of Novel 1-(Imidazo[1,2-a]pyridin-6-yl)pyridin-2(1H)-one Derivatives.
J Med Chem
; 59(3): 1116-39, 2016 Feb 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-26736071
12.
Correction to Melanin-Concentrating Hormone Receptor 1 Antagonists Lacking an Aliphatic Amine: Synthesis and Structure-Activity Relationships of Novel 1-(Imidazo[1,2-a]pyridin-6-yl)pyridin-2(1H)-one Derivatives.
J Med Chem
; 59(7): 3577, 2016 Apr 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-27045534
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