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Discovery of Selective Matriptase and Hepsin Serine Protease Inhibitors: Useful Chemical Tools for Cancer Cell Biology.
Damalanka, Vishnu C; Han, Zhenfu; Karmakar, Partha; O'Donoghue, Anthony J; La Greca, Florencia; Kim, Tommy; Pant, Shishir M; Helander, Jonathan; Klefström, Juha; Craik, Charles S; Janetka, James W.
Afiliación
  • Damalanka VC; Department of Biochemistry and Molecular Biophysics , Washington University School of Medicine , St. Louis , Missouri , 63110 , United States.
  • Han Z; Department of Biochemistry and Molecular Biophysics , Washington University School of Medicine , St. Louis , Missouri , 63110 , United States.
  • Karmakar P; Department of Biochemistry and Molecular Biophysics , Washington University School of Medicine , St. Louis , Missouri , 63110 , United States.
  • O'Donoghue AJ; Skaggs School of Pharmacy and Pharmaceutical Sciences , University of California , San Diego , California , 92093 , United States.
  • La Greca F; Department of Pharmaceutical Chemistry , University of California , San Francisco , California , 94158 , United States.
  • Kim T; Department of Pharmaceutical Chemistry , University of California , San Francisco , California , 94158 , United States.
  • Pant SM; Department of Biochemistry and Molecular Biophysics , Washington University School of Medicine , St. Louis , Missouri , 63110 , United States.
  • Helander J; Cancer Cell Circuitry Laboratory, Research Programs Unit/Translational Cancer Biology & Medicum , University of Helsinki , P.O. Box 63, Haartmaninkatu 8 , 00014 Helsinki , Finland.
  • Klefström J; Department of Biochemistry and Molecular Biophysics , Washington University School of Medicine , St. Louis , Missouri , 63110 , United States.
  • Craik CS; Cancer Cell Circuitry Laboratory, Research Programs Unit/Translational Cancer Biology & Medicum , University of Helsinki , P.O. Box 63, Haartmaninkatu 8 , 00014 Helsinki , Finland.
  • Janetka JW; Department of Pharmaceutical Chemistry , University of California , San Francisco , California , 94158 , United States.
J Med Chem ; 62(2): 480-490, 2019 01 24.
Article en En | MEDLINE | ID: mdl-30571119

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Serina Endopeptidasas / Inhibidores de Serina Proteinasa Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Serina Endopeptidasas / Inhibidores de Serina Proteinasa Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Estados Unidos