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Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors.
Hu, Jianping; Tian, Chang-Qing; Damaneh, Mohammadali Soleimani; Li, Yanlian; Cao, Danyan; Lv, Kaikai; Yu, Ting; Meng, Tao; Chen, Danqi; Wang, Xin; Chen, Lin; Li, Jian; Song, Shan-Shan; Huan, Xia-Juan; Qin, Lihuai; Shen, Jingkang; Wang, Ying-Qing; Miao, Ze-Hong; Xiong, Bing.
Afiliación
  • Hu J; University of Chinese Academy of Sciences , NO.19A Yuquan Road , Beijing 100049 , China.
  • Tian CQ; University of Chinese Academy of Sciences , NO.19A Yuquan Road , Beijing 100049 , China.
  • Damaneh MS; University of Chinese Academy of Sciences , NO.19A Yuquan Road , Beijing 100049 , China.
  • Lv K; University of Chinese Academy of Sciences , NO.19A Yuquan Road , Beijing 100049 , China.
  • Qin L; Center for Chemical Biology and Drug Discovery, Department of Pharmacological Sciences, Tisch Cancer Institute , Icahn School of Medicine at Mount Sinai , New York , New York 10029 , United States.
  • Wang YQ; University of Chinese Academy of Sciences , NO.19A Yuquan Road , Beijing 100049 , China.
  • Miao ZH; University of Chinese Academy of Sciences , NO.19A Yuquan Road , Beijing 100049 , China.
  • Xiong B; University of Chinese Academy of Sciences , NO.19A Yuquan Road , Beijing 100049 , China.
J Med Chem ; 62(18): 8642-8663, 2019 09 26.
Article en En | MEDLINE | ID: mdl-31490070

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Péptidos / Diseño de Fármacos / Proteínas Tipo de estudio: Prognostic_studies Límite: Animals / Humans / Male Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: China

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Péptidos / Diseño de Fármacos / Proteínas Tipo de estudio: Prognostic_studies Límite: Animals / Humans / Male Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: China