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Discovery of dihydroxyindole-2-carboxylic acid derivatives as dual allosteric HIV-1 Integrase and Reverse Transcriptase associated Ribonuclease H inhibitors.
Esposito, Francesca; Sechi, Mario; Pala, Nicolino; Sanna, Adele; Koneru, Pratibha Chowdary; Kvaratskhelia, Mamuka; Naesens, Lieve; Corona, Angela; Grandi, Nicole; di Santo, Roberto; D'Amore, Vincenzo Maria; Di Leva, Francesco Saverio; Novellino, Ettore; Cosconati, Sandro; Tramontano, Enzo.
Afiliación
  • Esposito F; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria SS554, 09042, Monserrato (CA), Italy. Electronic address: francescaesposito@unica.it.
  • Sechi M; Department of Chemistry and Pharmacy, University of Sassari, Via Vienna 2, 07100, Sassari, Italy.
  • Pala N; Department of Chemistry and Pharmacy, University of Sassari, Via Vienna 2, 07100, Sassari, Italy.
  • Sanna A; Department of Chemistry and Pharmacy, University of Sassari, Via Vienna 2, 07100, Sassari, Italy.
  • Koneru PC; Division of Infectious Diseases, University of Colorado School of Medicine, Aurora, CO, 80045, USA.
  • Kvaratskhelia M; Division of Infectious Diseases, University of Colorado School of Medicine, Aurora, CO, 80045, USA.
  • Naesens L; Rega Institute for Medical Research, KU Leuven, B-3000, Leuven, Belgium.
  • Corona A; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria SS554, 09042, Monserrato (CA), Italy.
  • Grandi N; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria SS554, 09042, Monserrato (CA), Italy.
  • di Santo R; Department of Drug Chemistry and Technologies, Istituto Pasteur-Fondazione Cenci Bolognetti, "Sapienza" Università di Roma, Roma, Italy.
  • D'Amore VM; Department of Pharmacy, University of Naples Federico II, Via D. Montesano 49, 80131, Naples, Italy.
  • Di Leva FS; Department of Pharmacy, University of Naples Federico II, Via D. Montesano 49, 80131, Naples, Italy.
  • Novellino E; Department of Pharmacy, University of Naples Federico II, Via D. Montesano 49, 80131, Naples, Italy.
  • Cosconati S; DiSTABiF, University of Campania Luigi Vanvitelli, Via Vivaldi, 43, 81100, Caserta, Italy.
  • Tramontano E; Department of Life and Environmental Sciences, University of Cagliari, Cittadella Universitaria SS554, 09042, Monserrato (CA), Italy.
Antiviral Res ; 174: 104671, 2020 02.
Article en En | MEDLINE | ID: mdl-31812637

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Ácidos Carboxílicos / VIH-1 / Inhibidores de Integrasa VIH / Ribonucleasa H del Virus de la Inmunodeficiencia Humana / Transcriptasa Inversa del VIH Tipo de estudio: Risk_factors_studies Límite: Humans Idioma: En Revista: Antiviral Res Año: 2020 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Ácidos Carboxílicos / VIH-1 / Inhibidores de Integrasa VIH / Ribonucleasa H del Virus de la Inmunodeficiencia Humana / Transcriptasa Inversa del VIH Tipo de estudio: Risk_factors_studies Límite: Humans Idioma: En Revista: Antiviral Res Año: 2020 Tipo del documento: Article