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1-(Piperidin-3-yl)thymine amides as inhibitors of M. tuberculosis thymidylate kinase.
Jian, Yanlin; Risseeuw, Martijn D P; Froeyen, Mathy; Song, Lijun; Cappoen, Davie; Cos, Paul; Munier-Lehmann, Hélène; van Calenbergh, Serge.
Afiliación
  • Jian Y; Laboratory for Medicinal Chemistry, Faculty of Pharmaceutical Sciences, Ghent University, Ghent, Belgium.
  • Risseeuw MDP; Laboratory for Medicinal Chemistry, Faculty of Pharmaceutical Sciences, Ghent University, Ghent, Belgium.
  • Froeyen M; Department of Medicinal Chemistry, Rega Institute for Medical Research, KU Leuven, Leuven, Belgium.
  • Song L; Laboratory for Medicinal Chemistry, Faculty of Pharmaceutical Sciences, Ghent University, Ghent, Belgium.
  • Cappoen D; Laboratory for Microbiology, Parasitology and Hygiene (LMPH), Department of Pharmaceutical Sciences, University of Antwerp, Antwerp, Belgium.
  • Cos P; Laboratory for Microbiology, Parasitology and Hygiene (LMPH), Department of Pharmaceutical Sciences, University of Antwerp, Antwerp, Belgium.
  • Munier-Lehmann H; Unit of Chemistry and Biocatalysis, Department of Structural Biology and Chemistry, Institut Pasteur, CNRS UMR3523, Paris, France.
  • van Calenbergh S; Laboratory for Medicinal Chemistry, Faculty of Pharmaceutical Sciences, Ghent University, Ghent, Belgium.
J Enzyme Inhib Med Chem ; 34(1): 1730-1739, 2019 Dec.
Article en En | MEDLINE | ID: mdl-31822127

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Timina / Nucleósido-Fosfato Quinasa / Inhibidores Enzimáticos / Amidas / Mycobacterium tuberculosis / Antituberculosos Tipo de estudio: Prognostic_studies Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Bélgica

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Timina / Nucleósido-Fosfato Quinasa / Inhibidores Enzimáticos / Amidas / Mycobacterium tuberculosis / Antituberculosos Tipo de estudio: Prognostic_studies Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Bélgica