1.
Bioorg Med Chem Lett
; 17(4): 974-7, 2007 Feb 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-17187980
RESUMEN
A novel class of 1H-(benzimidazol-2-yl)-1H-pyridin-2-one inhibitors of insulin-like growth factor I (IGF-1R) kinase is described. This report discusses the SAR of 4-(2-hydroxy-2-phenylethylamino)-substituted pyridones with improved IGF-1R potency.