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Discovery of Pyrazolopyridones as a Novel Class of Gyrase B Inhibitors Using Structure Guided Design.
Cross, Jason B; Zhang, Jing; Yang, Qingyi; Mesleh, Michael F; Romero, Jan Antoinette C; Wang, Bin; Bevan, Doug; Poutsiaka, Katherine M; Epie, Felix; Moy, Terence; Daniel, Anu; Shotwell, Joseph; Chamberlain, Brian; Carter, Nicole; Andersen, Ole; Barker, John; Ryan, M Dominic; Metcalf, Chester A; Silverman, Jared; Nguyen, Kien; Lippa, Blaise; Dolle, Roland E.
Afiliación
  • Cross JB; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Zhang J; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Yang Q; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Mesleh MF; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Romero JA; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Wang B; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Bevan D; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Poutsiaka KM; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Epie F; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Moy T; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Daniel A; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Shotwell J; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Chamberlain B; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Carter N; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Andersen O; Evotec U.K., Ltd. , 114 Innovation Drive, Milton Park, Abingdon, Oxfordshire OX14 4RZ, United Kingdom.
  • Barker J; Evotec U.K., Ltd. , 114 Innovation Drive, Milton Park, Abingdon, Oxfordshire OX14 4RZ, United Kingdom.
  • Ryan MD; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Metcalf CA; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Silverman J; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Nguyen K; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Lippa B; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
  • Dolle RE; Cubist Pharmaceuticals, Inc. , 65 Hayden Avenue, Lexington, Massachusetts 02421, United States.
ACS Med Chem Lett ; 7(4): 374-8, 2016 Apr 14.
Article en En | MEDLINE | ID: mdl-27096044

Texto completo: 1 Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2016 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Base de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2016 Tipo del documento: Article País de afiliación: Estados Unidos