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X-ray structures of endothelin ETB receptor bound to clinical antagonist bosentan and its analog.
Shihoya, Wataru; Nishizawa, Tomohiro; Yamashita, Keitaro; Inoue, Asuka; Hirata, Kunio; Kadji, Francois Marie Ngako; Okuta, Akiko; Tani, Kazutoshi; Aoki, Junken; Fujiyoshi, Yoshinori; Doi, Tomoko; Nureki, Osamu.
Afiliación
  • Shihoya W; Department of Basic Medicinal Sciences, Graduate School of Pharmaceutical Sciences, Nagoya University, Nagoya, Japan.
  • Nishizawa T; Cellular and Structural Physiology Institute, Nagoya University, Nagoya, Japan.
  • Yamashita K; Department of Biophysics and Biochemistry, Graduate School of Science, The University of Tokyo, Tokyo, Japan.
  • Inoue A; Department of Biophysics and Biochemistry, Graduate School of Science, The University of Tokyo, Tokyo, Japan.
  • Hirata K; Precursory Research for Embryonic Science and Technology (PRESTO), Japan Science and Technology Agency, Kawaguchi, Japan.
  • Kadji FMN; RIKEN SPring-8 Center, Sayo, Japan.
  • Okuta A; Precursory Research for Embryonic Science and Technology (PRESTO), Japan Science and Technology Agency, Kawaguchi, Japan.
  • Tani K; Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan.
  • Aoki J; Precursory Research for Embryonic Science and Technology (PRESTO), Japan Science and Technology Agency, Kawaguchi, Japan.
  • Fujiyoshi Y; RIKEN SPring-8 Center, Sayo, Japan.
  • Doi T; Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Japan.
  • Nureki O; Cellular and Structural Physiology Institute, Nagoya University, Nagoya, Japan.
Nat Struct Mol Biol ; 24(9): 758-764, 2017 Sep.
Article en En | MEDLINE | ID: mdl-28805809

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Sulfonamidas / Receptor de Endotelina B / Antagonistas de los Receptores de Endotelina Límite: Humans Idioma: En Revista: Nat Struct Mol Biol Asunto de la revista: BIOLOGIA MOLECULAR Año: 2017 Tipo del documento: Article País de afiliación: Japón

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Sulfonamidas / Receptor de Endotelina B / Antagonistas de los Receptores de Endotelina Límite: Humans Idioma: En Revista: Nat Struct Mol Biol Asunto de la revista: BIOLOGIA MOLECULAR Año: 2017 Tipo del documento: Article País de afiliación: Japón