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Novel and Selective TLR7 Antagonists among the Imidazo[1,2-a]pyrazines, Imidazo[1,5-a]quinoxalines, and Pyrazolo[1,5-a]quinoxalines Series.
Bou Karroum, Nour; Moarbess, Georges; Guichou, Jean-François; Bonnet, Pierre-Antoine; Patinote, Cindy; Bouharoun-Tayoun, Hasnaa; Chamat, Soulaima; Cuq, Pierre; Diab-Assaf, Mona; Kassab, Issam; Deleuze-Masquefa, Carine.
Afiliación
  • Bou Karroum N; Institut des Biomolécules Max Mousseron (IBMM), UMR 5247 F16, CNRS, Université de Montpellier , Faculté de Pharmacie , 15 avenue Charles Flahault , BP 14491, Montpellier 34093 Cedex 5 , France.
  • Moarbess G; Tumorigenèse et Pharmacologie Antitumorale , Lebanese University, EDST , BP 90656, Fanar Jdeideh 1202 , Lebanon.
  • Guichou JF; Tumorigenèse et Pharmacologie Antitumorale , Lebanese University, EDST , BP 90656, Fanar Jdeideh 1202 , Lebanon.
  • Bonnet PA; CNRS, UMR 5048, INSERM, U105, Université de Montpellier, Centre de Biochimie Structurale , Montpellier F-34090 , France.
  • Patinote C; Institut des Biomolécules Max Mousseron (IBMM), UMR 5247 F16, CNRS, Université de Montpellier , Faculté de Pharmacie , 15 avenue Charles Flahault , BP 14491, Montpellier 34093 Cedex 5 , France.
  • Bouharoun-Tayoun H; Institut des Biomolécules Max Mousseron (IBMM), UMR 5247 F16, CNRS, Université de Montpellier , Faculté de Pharmacie , 15 avenue Charles Flahault , BP 14491, Montpellier 34093 Cedex 5 , France.
  • Chamat S; Laboratory of Immunology and Vector-Borne Diseases, Faculty of Public Health , Lebanese University , Fanar Jdeideh 1202 , Lebanon.
  • Cuq P; Laboratory of Immunology and Vector-Borne Diseases, Faculty of Public Health , Lebanese University , Fanar Jdeideh 1202 , Lebanon.
  • Diab-Assaf M; Faculty of Medical Sciences , Lebanese University , Hadath 1500 , Lebanon.
  • Kassab I; Institut des Biomolécules Max Mousseron (IBMM), UMR 5247 F16, CNRS, Université de Montpellier , Faculté de Pharmacie , 15 avenue Charles Flahault , BP 14491, Montpellier 34093 Cedex 5 , France.
  • Deleuze-Masquefa C; Tumorigenèse et Pharmacologie Antitumorale , Lebanese University, EDST , BP 90656, Fanar Jdeideh 1202 , Lebanon.
J Med Chem ; 62(15): 7015-7031, 2019 08 08.
Article en En | MEDLINE | ID: mdl-31283223

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Pirazinas / Quinoxalinas / Receptor Toll-Like 7 / Imidazoles Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Francia

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Pirazinas / Quinoxalinas / Receptor Toll-Like 7 / Imidazoles Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Francia