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Structure-Based Design of Y-Shaped Covalent TEAD Inhibitors.
Lu, Wenchao; Fan, Mengyang; Ji, Wenzhi; Tse, Jason; You, Inchul; Ficarro, Scott B; Tavares, Isidoro; Che, Jianwei; Kim, Audrey Y; Zhu, Xijun; Boghossian, Andrew; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Hinshaw, Stephen M; Nabet, Behnam; Corsello, Steven M; Kwiatkowski, Nicholas; Marto, Jarrod A; Zhang, Tinghu; Gray, Nathanael S.
Afiliación
  • Lu W; Department of Chemical and Systems Biology, Chem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States.
  • Fan M; Hangzhou Institute of Medicine (HIM), Chinese Academy of Sciences, Hangzhou, Zhejiang 310022, China.
  • Ji W; Department of Chemical and Systems Biology, Chem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States.
  • Tse J; Department of Chemical and Systems Biology, Chem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States.
  • You I; Department of Chemical and Systems Biology, Chem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States.
  • Ficarro SB; Department of Cancer Biology, Blais Proteomics Center, Center for Emergent Drug Targets, Dana-Farber Cancer Institute, Boston, Massachusetts 02215, United States.
  • Tavares I; Department of Cancer Biology, Blais Proteomics Center, Center for Emergent Drug Targets, Dana-Farber Cancer Institute, Boston, Massachusetts 02215, United States.
  • Che J; Center for Protein Degradation, Dana-Farber Cancer Institute, Boston, Massachusetts 02215, United States.
  • Kim AY; Department of Chemical and Systems Biology, Chem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States.
  • Zhu X; Department of Chemistry, Stanford University, Stanford, California 94305, United States.
  • Boghossian A; Broad Institute of MIT and Harvard, Cambridge, Massachusetts 02142, United States.
  • Rees MG; Broad Institute of MIT and Harvard, Cambridge, Massachusetts 02142, United States.
  • Ronan MM; Broad Institute of MIT and Harvard, Cambridge, Massachusetts 02142, United States.
  • Roth JA; Broad Institute of MIT and Harvard, Cambridge, Massachusetts 02142, United States.
  • Hinshaw SM; Department of Chemical and Systems Biology, Chem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States.
  • Nabet B; Human Biology Division, Fred Hutchinson Cancer Center, Seattle, Washington 98109, United States.
  • Corsello SM; Department of Medicine and Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States.
  • Kwiatkowski N; Center for Protein Degradation, Dana-Farber Cancer Institute, Boston, Massachusetts 02215, United States.
  • Marto JA; Department of Cancer Biology, Blais Proteomics Center, Center for Emergent Drug Targets, Dana-Farber Cancer Institute, Boston, Massachusetts 02215, United States.
  • Zhang T; Department of Pathology, Brigham and Women's Hospital and Harvard Medical School, Boston, Massachusetts 02215, United States.
  • Gray NS; Department of Chemical and Systems Biology, Chem-H and Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States.
J Med Chem ; 66(7): 4617-4632, 2023 04 13.
Article en En | MEDLINE | ID: mdl-36946421

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Proteínas de Unión al ADN / Neoplasias Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Proteínas de Unión al ADN / Neoplasias Límite: Animals / Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos