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Discovery of Guanfacine as a Novel TAAR1 Agonist: A Combination Strategy through Molecular Modeling Studies and Biological Assays.
Cichero, Elena; Francesconi, Valeria; Casini, Beatrice; Casale, Monica; Kanov, Evgeny; Gerasimov, Andrey S; Sukhanov, Ilya; Savchenko, Artem; Espinoza, Stefano; Gainetdinov, Raul R; Tonelli, Michele.
Afiliación
  • Cichero E; Department of Pharmacy, Section of Medicinal Chemistry, School of Medical and Pharmaceutical Sciences, University of Genoa, 16132 Genoa, Italy.
  • Francesconi V; Department of Pharmacy, Section of Medicinal Chemistry, School of Medical and Pharmaceutical Sciences, University of Genoa, 16132 Genoa, Italy.
  • Casini B; Department of Pharmacy, Section of Medicinal Chemistry, School of Medical and Pharmaceutical Sciences, University of Genoa, 16132 Genoa, Italy.
  • Casale M; Section of Chemistry and Food and Pharmaceutical Technologies, University of Genoa, 16148 Genoa, Italy.
  • Kanov E; Institute of Translational Biomedicine, St. Petersburg State University, 199034 St. Petersburg, Russia.
  • Gerasimov AS; St. Petersburg University Hospital, St. Petersburg State University, 199034 St. Petersburg, Russia.
  • Sukhanov I; Institute of Translational Biomedicine, St. Petersburg State University, 199034 St. Petersburg, Russia.
  • Savchenko A; Valdman Institute of Pharmacology, Pavlov First St. Petersburg State Medical University, 197022 St. Petersburg, Russia.
  • Espinoza S; Valdman Institute of Pharmacology, Pavlov First St. Petersburg State Medical University, 197022 St. Petersburg, Russia.
  • Gainetdinov RR; Department of Health Sciences and Research Center on Autoimmune and Allergic Diseases (CAAD), University of Piemonte Orientale (UPO), 28100 Novara, Italy.
  • Tonelli M; Central RNA Laboratory, Istituto Italiano di Tecnologia (IIT), 16152 Genova, Italy.
Pharmaceuticals (Basel) ; 16(11)2023 Nov 20.
Article en En | MEDLINE | ID: mdl-38004497

Texto completo: 1 Base de datos: MEDLINE Idioma: En Revista: Pharmaceuticals (Basel) Año: 2023 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Base de datos: MEDLINE Idioma: En Revista: Pharmaceuticals (Basel) Año: 2023 Tipo del documento: Article País de afiliación: Italia