Detalhe da pesquisa
1.
First-in-human study of alpibectir (BVL-GSK098), a novel potent anti-TB drug.
J Antimicrob Chemother
; 79(6): 1353-1361, 2024 Jun 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-38656557
2.
Short-course combination treatment for experimental chronic Chagas disease.
Sci Transl Med
; 15(726): eadg8105, 2023 12 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-38091410
3.
DNDI-6174 is a preclinical candidate for visceral leishmaniasis that targets the cytochrome bc1.
Sci Transl Med
; 15(726): eadh9902, 2023 12 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-38091406
4.
The small-molecule SMARt751 reverses Mycobacterium tuberculosis resistance to ethionamide in acute and chronic mouse models of tuberculosis.
Sci Transl Med
; 14(643): eaaz6280, 2022 05 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-35507672
5.
Identification of ß-Lactams Active against Mycobacterium tuberculosis by a Consortium of Pharmaceutical Companies and Academic Institutions.
ACS Infect Dis
; 8(3): 557-573, 2022 03 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-35192346
6.
Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents.
PLoS Negl Trop Dis
; 13(2): e0007129, 2019 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-30735501
7.
Hundreds of dual-stage antimalarial molecules discovered by a functional gametocyte screen.
Nat Commun
; 8: 15160, 2017 05 17.
Artigo
em Inglês
| MEDLINE | ID: mdl-28513586
8.
The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold.
J Med Chem
; 60(16): 6880-6896, 2017 08 24.
Artigo
em Inglês
| MEDLINE | ID: mdl-28806082
9.
Hit-to-Lead Optimization of a Novel Class of Potent, Broad-Spectrum Trypanosomacides.
J Med Chem
; 59(21): 9686-9720, 2016 11 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-27548560
10.
Carbamoyl Triazoles, Known Serine Protease Inhibitors, Are a Potent New Class of Antimalarials.
J Med Chem
; 58(16): 6448-55, 2015 Aug 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-26222445
11.
A Developability-Focused Optimization Approach Allows Identification of in Vivo Fast-Acting Antimalarials: N-[3-[(Benzimidazol-2-yl)amino]propyl]amides.
J Med Chem
; 58(11): 4573-80, 2015 Jun 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-25906200
12.
Correction to The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold.
J Med Chem
; 60(23): 9911, 2017 12 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-29164877