Detalhe da pesquisa
1.
Phase Separation of Disease-Associated SHP2 Mutants Underlies MAPK Hyperactivation.
Cell
; 183(2): 490-502.e18, 2020 10 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-33002410
2.
Small molecule approaches to treat autoimmune and inflammatory diseases (Part I): Kinase inhibitors.
Bioorg Med Chem Lett
; 38: 127862, 2021 04 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-33609659
3.
Small molecule approaches to treat autoimmune and inflammatory diseases (Part III): Targeting cytokines and cytokine receptor complexes.
Bioorg Med Chem Lett
; 48: 128229, 2021 09 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-34214508
4.
Intramolecular N-Me and N-H aminoetherification for the synthesis of N-unprotected 3-amino-O-heterocycles.
Org Biomol Chem
; 19(3): 557-560, 2021 01 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-33399609
5.
Highly Chemo- and Regioselective Vinylation of N-Heteroarenes with Vinylsulfonium Salts.
J Org Chem
; 83(15): 8627-8635, 2018 Aug 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-29799743
6.
Palladium-Catalyzed Difluoromethylation of Aryl Chlorides and Triflates and Its Applications in the Preparation of Difluoromethylated Derivatives of Drug/Agrochemical Molecules.
J Org Chem
; 83(2): 1077-1083, 2018 01 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-29271195
7.
Potassium Iodide-Promoted One-Pot Synthesis of Fluoroalkylated Quinoxalines via a Tandem Michael Addition/Azidation/Cycloamination Approach.
J Org Chem
; 83(16): 9422-9429, 2018 08 17.
Artigo
em Inglês
| MEDLINE | ID: mdl-30025451
8.
C-H Bond Functionalization of Tetrahydropyridopyrimidines and Other Related Hetereocycles.
J Org Chem
; 82(24): 13678-13685, 2017 12 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-29134810
9.
Divergent copper-mediated dimerization and hydroxylation of benzamides involving C-H bond functionalization.
Org Biomol Chem
; 14(18): 4239-46, 2016 May 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-27073988
10.
Mineralocorticoid receptor antagonists: identification of heterocyclic amide replacements in the oxazolidinedione series.
Bioorg Med Chem Lett
; 24(7): 1681-4, 2014 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-24630411
11.
Discovery of novel oxazolidinedione derivatives as potent and selective mineralocorticoid receptor antagonists.
Bioorg Med Chem Lett
; 23(15): 4388-92, 2013 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23777778
12.
Gold-catalyzed formation of heterocycles - an enabling new technology for medicinal chemistry.
Drug Discov Today Technol
; 10(1): e3-14, 2013.
Artigo
em Inglês
| MEDLINE | ID: mdl-24050224
13.
Discovery of Linvencorvir (RG7907), a Hepatitis B Virus Core Protein Allosteric Modulator, for the Treatment of Chronic HBV Infection.
J Med Chem
; 66(6): 4253-4270, 2023 03 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-36896968
14.
Discovery of 4,5,6,7-Tetrahydropyrazolo[1.5-a]pyrizine Derivatives as Core Protein Allosteric Modulators (CpAMs) for the Inhibition of Hepatitis B Virus.
J Med Chem
; 66(20): 14116-14132, 2023 10 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-37801325
15.
The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors.
Bioorg Med Chem Lett
; 22(1): 658-65, 2012 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-22079761
16.
Discovery of benzodihydroisofurans as novel, potent, bioavailable and brain-penetrant prolylcarboxypeptidase inhibitors.
Bioorg Med Chem Lett
; 22(4): 1550-6, 2012 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22264488
17.
Translation Potential and Challenges of In Vitro and Murine Models in Cancer Clinic.
Cells
; 11(23)2022 Nov 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-36497126
18.
Discovery of Novel cccDNA Reducers toward the Cure of Hepatitis B Virus Infection.
J Med Chem
; 65(16): 10938-10955, 2022 08 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-35973101
19.
Discovery of benzimidazole pyrrolidinyl amides as prolylcarboxypeptidase inhibitors.
Bioorg Med Chem Lett
; 21(5): 1299-305, 2011 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21315588
20.
Discovery of pyrazolyl propionyl cyclohexenamide derivatives as full agonists for the high affinity niacin receptor GPR109A.
Bioorg Med Chem Lett
; 20(11): 3372-5, 2010 Jun 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20452209