Detalhe da pesquisa
1.
Stereodivergent Synthesis of Biologically Active Spironucleoside Scaffolds via Catalytic Cyclopropanation of 4-exo-Methylene Furanosides.
J Org Chem
; 86(23): 17344-17361, 2021 12 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-34748342
2.
Synthesis and Reactivity of Spirocarbocycles as Scaffolds for Nucleoside Analogues.
J Org Chem
; 85(23): 14989-15005, 2020 12 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-33196210
3.
Stereoselective Reductions of 3-Substituted Cyclobutanones: A Comparison between Experiment and Theory.
J Org Chem
; 85(12): 7803-7816, 2020 06 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-32441520
4.
Towards the Design of Optically Active Thiophene S-Oxides using Quantum Chemistry.
Chemistry
; 25(11): 2840-2851, 2019 Feb 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-30600854
5.
Preparation of 4'-Spirocyclobutyl Nucleoside Analogues as Novel and Versatile Adenosine Scaffolds.
Chemistry
; 25(67): 15419-15423, 2019 Dec 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-31609050
6.
The 1,3-diyne linker as a rigid "i,i+7" staple for α-helix stabilization: Stereochemistry at work.
J Pept Sci
; 25(7): e3194, 2019 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-31215108
7.
The antibacterial prodrug activator Rv2466c is a mycothiol-dependent reductase in the oxidative stress response of Mycobacterium tuberculosis.
J Biol Chem
; 292(32): 13097-13110, 2017 08 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-28620052
8.
Metal-Free Cyclization of ortho-Nitroaryl Ynamides and Ynamines towards Spiropseudoindoxyls.
Angew Chem Int Ed Engl
; 57(20): 5660-5664, 2018 05 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-29570239
9.
Synthesis of 2-Fluoro-1,4-benzoxazines and 2-Fluoro-1,4-benzoxazepin-5-ones by Exploring the Nucleophilic Vinylic Substitution (S(N)V) Reaction of gem-Difluoroenamides.
J Org Chem
; 80(10): 5111-24, 2015 May 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-25901523
10.
Nucleophile-directed selective transformation of cis-1-tosyl-2-tosyloxymethyl-3-(trifluoromethyl)aziridine into aziridines, azetidines, and benzo-fused dithianes, oxathianes, dioxanes, and (thio)morpholines.
Chemistry
; 19(19): 5966-71, 2013 May 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-23512331
11.
Synthesis of 1-alkyl-2-(trifluoromethyl)azetidines and their regiospecific ring opening toward diverse α-(trifluoromethyl)amines via intermediate azetidinium salts.
J Org Chem
; 77(14): 5982-92, 2012 Jul 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-22721444
12.
Synthesis of 3-amino-4-fluoropyrazoles.
J Org Chem
; 76(10): 4105-11, 2011 May 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-21500813
13.
Straightforward synthesis of 1-alkyl-2-(trifluoromethyl)aziridines starting from 1,1,1-trifluoroacetone.
Org Biomol Chem
; 9(20): 7217-23, 2011 Oct 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-21874207
14.
Regio- and Stereoselective Synthesis of C-4' Spirocyclobutyl Ribofuranose Scaffolds and Their Use as Biologically Active Nucleoside Analogues.
Org Lett
; 23(22): 8828-8833, 2021 11 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-34730365
15.
Short synthesis of the seed germination inhibitor 3,4,5-trimethyl-2(5H)-furanone.
J Org Chem
; 75(16): 5750-3, 2010 Aug 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-20704450
16.
Heteroaryl cross-coupling as an entry toward the synthesis of lavendamycin analogues: a model study.
J Org Chem
; 75(2): 424-33, 2010 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20017470
17.
Improved Arndt-Eistert synthesis of alpha-diazoketones requiring minimal diazomethane in the presence of calcium oxide as acid scavenger.
J Org Chem
; 75(16): 5760-3, 2010 Aug 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-20672806
18.
Synthesis of 4-substituted 3,3-difluoropiperidines.
J Org Chem
; 75(3): 929-32, 2010 Feb 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-20050617
19.
Synthesis of 5-amino- and 5-hydroxy-3,3-difluoropiperidines.
Org Biomol Chem
; 8(20): 4514-7, 2010 Oct 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-20668779
20.
Synthesis of aminomethylated 4-fluoropiperidines and 3-fluoropyrrolidines.
Org Biomol Chem
; 8(11): 2509-12, 2010 Jun 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-20407687