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Design, synthesis, molecular docking and 3D-QSAR studies of potent inhibitors of enoyl-acyl carrier protein reductase as potential antimycobacterial agents.
More, Uttam A; Joshi, Shrinivas D; Aminabhavi, Tejraj M; Gadad, Andanappa K; Nadagouda, Mallikarjuna N; Kulkarni, Venkatrao H.
Afiliação
  • More UA; Novel Drug Design and Discovery Laboratory, Department of Pharmaceutical Chemistry, S.E.T's College of Pharmacy, Sangolli Rayanna Nagar, Dharwad 580 002, India; Centre for Research and Development, Prist University, Thanjavur 613 403, Tamil Nadu, India.
  • Joshi SD; Novel Drug Design and Discovery Laboratory, Department of Pharmaceutical Chemistry, S.E.T's College of Pharmacy, Sangolli Rayanna Nagar, Dharwad 580 002, India. Electronic address: shrinivasdj@rediffmail.com.
  • Aminabhavi TM; Novel Drug Design and Discovery Laboratory, Department of Pharmaceutical Chemistry, S.E.T's College of Pharmacy, Sangolli Rayanna Nagar, Dharwad 580 002, India.
  • Gadad AK; School of Pharmacy, Faculty of Medical Sciences (The University of the West Indies, St. Augustine), Champs-Fleurs, Mount-Hope, Trinidad and Tobago.
  • Nadagouda MN; Novel Drug Design and Discovery Laboratory, Department of Pharmaceutical Chemistry, S.E.T's College of Pharmacy, Sangolli Rayanna Nagar, Dharwad 580 002, India.
  • Kulkarni VH; Novel Drug Design and Discovery Laboratory, Department of Pharmaceutical Chemistry, S.E.T's College of Pharmacy, Sangolli Rayanna Nagar, Dharwad 580 002, India.
Eur J Med Chem ; 71: 199-218, 2014 Jan.
Article em En | MEDLINE | ID: mdl-24292339

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oxirredutases / Proteínas de Bactérias / Desenho de Fármacos / Hidrazonas / Antibacterianos / Mycobacterium tuberculosis Idioma: En Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Índia

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oxirredutases / Proteínas de Bactérias / Desenho de Fármacos / Hidrazonas / Antibacterianos / Mycobacterium tuberculosis Idioma: En Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Índia