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Synthesis, modification and docking studies of 5-sulfonyl isatin derivatives as SARS-CoV 3C-like protease inhibitors.
Liu, Wei; Zhu, He-Min; Niu, Guo-Jun; Shi, En-Zhi; Chen, Jie; Sun, Bo; Chen, Wei-Qiang; Zhou, Hong-Gang; Yang, Cheng.
Afiliação
  • Liu W; College of Sciences, Tianjin University of Science and Technology, Tianjin 300457, China. Electronic address: liuwei2006@tust.edu.cn.
  • Zhu HM; College of Life Sciences, NanKai University, Tianjin 300071, China.
  • Niu GJ; High Throughput Molecular Drug Discovery Center, Tianjin International Joint Academy of Biotechnology and Medicine, TEDA, Tianjin 300457, China.
  • Shi EZ; College of Life Sciences, NanKai University, Tianjin 300071, China.
  • Chen J; College of Pharmacy, NanKai University, Tianjin 300071, China.
  • Sun B; High Throughput Molecular Drug Discovery Center, Tianjin International Joint Academy of Biotechnology and Medicine, TEDA, Tianjin 300457, China.
  • Chen WQ; High Throughput Molecular Drug Discovery Center, Tianjin International Joint Academy of Biotechnology and Medicine, TEDA, Tianjin 300457, China.
  • Zhou HG; College of Pharmacy, NanKai University, Tianjin 300071, China.
  • Yang C; College of Pharmacy, NanKai University, Tianjin 300071, China; High Throughput Molecular Drug Discovery Center, Tianjin International Joint Academy of Biotechnology and Medicine, TEDA, Tianjin 300457, China.
Bioorg Med Chem ; 22(1): 292-302, 2014 Jan 01.
Article em En | MEDLINE | ID: mdl-24316352

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Proteases / Coronavírus Relacionado à Síndrome Respiratória Aguda Grave / Isatina Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Proteases / Coronavírus Relacionado à Síndrome Respiratória Aguda Grave / Isatina Idioma: En Ano de publicação: 2014 Tipo de documento: Article