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GW779439X and Its Pyrazolopyridazine Derivatives Inhibit the Serine/Threonine Kinase Stk1 and Act As Antibiotic Adjuvants against ß-Lactam-Resistant Staphylococcus aureus.
Schaenzer, Adam J; Wlodarchak, Nathan; Drewry, David H; Zuercher, William J; Rose, Warren E; Ferrer, Carla A; Sauer, John-Demian; Striker, Rob.
Afiliação
  • Schaenzer AJ; Department of Medical Microbiology and Immunology , University of Wisconsin-Madison , 1550 Linden Drive , Madison , Wisconsin 53706 , United States.
  • Wlodarchak N; Department of Medicine , University of Wisconsin-Madison , 1685 Highland Avenue , Madison , Wisconsin 53706 , United States.
  • Drewry DH; Department of Medical Microbiology and Immunology , University of Wisconsin-Madison , 1550 Linden Drive , Madison , Wisconsin 53706 , United States.
  • Zuercher WJ; Department of Medicine , University of Wisconsin-Madison , 1685 Highland Avenue , Madison , Wisconsin 53706 , United States.
  • Rose WE; UNC Eshelman School of Pharmacy, SGC Center for Chemical Biology , University of North Carolina at Chapel Hill , 120 Mason Farm Road , Chapel Hill , North Carolina 27599 , United States.
  • Ferrer CA; UNC Eshelman School of Pharmacy, SGC Center for Chemical Biology , University of North Carolina at Chapel Hill , 120 Mason Farm Road , Chapel Hill , North Carolina 27599 , United States.
  • Sauer JD; Department of Medicine , University of Wisconsin-Madison , 1685 Highland Avenue , Madison , Wisconsin 53706 , United States.
  • Striker R; School of Pharmacy , University of Wisconsin-Madison , 777 Highland Avenue , Madison , Wisconsin 53705 , United States.
ACS Infect Dis ; 4(10): 1508-1518, 2018 10 12.
Article em En | MEDLINE | ID: mdl-30059625

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oxacilina / Piridazinas / Cefalosporinas / Adjuvantes Farmacêuticos / Resistência beta-Lactâmica / Inibidores de Proteínas Quinases / Tirosina Quinase 3 Semelhante a fms Idioma: En Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oxacilina / Piridazinas / Cefalosporinas / Adjuvantes Farmacêuticos / Resistência beta-Lactâmica / Inibidores de Proteínas Quinases / Tirosina Quinase 3 Semelhante a fms Idioma: En Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Estados Unidos