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Novel inhibitors of As(III) S-adenosylmethionine methyltransferase (AS3MT) identified by virtual screening.
Bürli, Roland W; Wei, Huijun; Ernst, Glen; Mariga, Abigail; Hardern, Ian M; Herlihy, Kara; Cross, Alan J; Wesolowski, Steven S; Chen, Hongming; McKay, Ronald D G; Weinberger, Daniel R; Brandon, Nicholas J; Barrow, James C.
Afiliação
  • Bürli RW; Neuroscience, IMED Biotech Unit, AstraZeneca, Cambridge CB21 6GH, UK. Electronic address: roland.burli@azneuro.com.
  • Wei H; Lieber Institute for Brain Development, 855 North Wolfe Street, Baltimore, MD 21205, USA.
  • Ernst G; Lieber Institute for Brain Development, 855 North Wolfe Street, Baltimore, MD 21205, USA.
  • Mariga A; Lieber Institute for Brain Development, 855 North Wolfe Street, Baltimore, MD 21205, USA.
  • Hardern IM; Discovery Sciences, IMED Biotech Unit, AstraZeneca, Cambridge CB4 0WG, UK.
  • Herlihy K; Discovery Sciences, IMED Biotech Unit, AstraZeneca, Cambridge CB4 0WG, UK.
  • Cross AJ; Neuroscience, IMED Biotech Unit, AstraZeneca Boston, Waltham, MA 02451, USA.
  • Wesolowski SS; Neuroscience, IMED Biotech Unit, AstraZeneca Boston, Waltham, MA 02451, USA.
  • Chen H; Discovery Sciences, IMED Biotech Unit, AstraZeneca Gothenburg, S-43183 Mölndal, Sweden.
  • McKay RDG; Lieber Institute for Brain Development, 855 North Wolfe Street, Baltimore, MD 21205, USA.
  • Weinberger DR; Lieber Institute for Brain Development, 855 North Wolfe Street, Baltimore, MD 21205, USA; Departments of Psychiatry, Neurology, Neuroscience and the McKusick-Nathans Institute of Genetic Medicine, Johns Hopkins University School of Medicine, Baltimore, MD 21287, USA.
  • Brandon NJ; Neuroscience, IMED Biotech Unit, AstraZeneca Boston, Waltham, MA 02451, USA.
  • Barrow JC; Lieber Institute for Brain Development, 855 North Wolfe Street, Baltimore, MD 21205, USA; Department of Pharmacology, Johns Hopkins University School of Medicine, 855 North Wolfe Street, Baltimore, MD 21287, USA. Electronic address: james.barrow@libd.org.
Bioorg Med Chem Lett ; 28(19): 3231-3235, 2018 10 15.
Article em En | MEDLINE | ID: mdl-30170942

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores Enzimáticos / Metiltransferases Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores Enzimáticos / Metiltransferases Idioma: En Ano de publicação: 2018 Tipo de documento: Article