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Design, synthesis and biological evaluation of novel human monoamine oxidase B inhibitors based on a fragment in an X-ray crystal structure.
Cheng, Kai; Li, Shiyu; Lv, Xiao; Tian, Yongbin; Kong, Haiyan; Huang, Xufeng; Duan, Yajun; Han, Jihong; Xie, Zhouling; Liao, Chenzhong.
Afiliação
  • Cheng K; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China.
  • Li S; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China.
  • Lv X; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China.
  • Tian Y; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China.
  • Kong H; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China.
  • Huang X; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China.
  • Duan Y; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China.
  • Han J; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China.
  • Xie Z; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China. Electronic address: zhoulingxie@hfut.edu.cn.
  • Liao C; School of Food and Biological Engineering, Hefei University of Technology, Hefei, Anhui 230009, PR China. Electronic address: czliao@hfut.edu.cn.
Bioorg Med Chem Lett ; 29(8): 1012-1018, 2019 04 15.
Article em En | MEDLINE | ID: mdl-30792039

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Monoaminoxidase / Inibidores da Monoaminoxidase Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Monoaminoxidase / Inibidores da Monoaminoxidase Idioma: En Ano de publicação: 2019 Tipo de documento: Article