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Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target Investigation.
Venugopala, Katharigatta N; Ramachandra, Pushpalatha; Tratrat, Christophe; Gleiser, Raquel M; Bhandary, Subhrajyoti; Chopra, Deepak; Morsy, Mohamed A; Aldhubiab, Bandar E; Attimarad, Mahesh; Nair, Anroop B; Sreeharsha, Nagaraja; Venugopala, Rashmi; Deb, Pran Kishore; Chandrashekharappa, Sandeep; Khalil, Hany Ezzat; Alwassil, Osama I; Abed, Sara Nidal; Bataineh, Yazan A; Palenge, Ramachandra; Haroun, Michelyne; Pottathil, Shinu; Girish, Meravanige B; Akrawi, Sabah H; Mohanlall, Viresh.
Afiliação
  • Venugopala KN; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Ramachandra P; Department of Biotechnology and Food Technology, Durban University of Technology, Durban 4001, South Africa.
  • Tratrat C; Department of Chemistry, School of Applied Sciences, REVA University, Bangalore 560 064, India.
  • Gleiser RM; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Bhandary S; CREAN-IMBIV (UNC-CONICET), Av. Valparaíso s.n., Córdoba, Argentina and FCEFyN, AV. Sarsfield 299, Universidad Nacional de Cordoba, Cordoba 5000, Argentina.
  • Chopra D; Department of Chemistry, Indian Institute of Science Education and Research Bhopal, Bhopal By-pass Road, Bhauri, Bhopal 462 066, Madhya Pradesh, India.
  • Morsy MA; Department of Chemistry, Indian Institute of Science Education and Research Bhopal, Bhopal By-pass Road, Bhauri, Bhopal 462 066, Madhya Pradesh, India.
  • Aldhubiab BE; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Attimarad M; Department of Pharmacology, Faculty of Medicine, Minia University, El-Minia 61511, Egypt.
  • Nair AB; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Sreeharsha N; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Venugopala R; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Deb PK; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Chandrashekharappa S; Department of Public Health Medicine, University of KwaZulu-Natal, Howard College Campus, Durban 4001, South Africa.
  • Khalil HE; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan.
  • Alwassil OI; Institute for Stem Cell Biology and Regenerative Medicine, NCBS, TIFR, GKVK, Bellary Road, Bangalore 560 065, India.
  • Abed SN; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Bataineh YA; Department of Pharmacognosy, Faculty of Pharmacy, Minia University, Minia 61519, Egypt.
  • Palenge R; Department of Pharmaceutical Sciences, College of Pharmacy, King Saud bin Abdulaziz University for Health Sciences, Riyadh 11481, Saudi Arabia.
  • Haroun M; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan.
  • Pottathil S; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan.
  • Girish MB; Department of Chemistry, School of Applied Sciences, REVA University, Bangalore 560 064, India.
  • Akrawi SH; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
  • Mohanlall V; Department of Biomedical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.
Molecules ; 25(6)2020 Mar 13.
Article em En | MEDLINE | ID: mdl-32183140

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Quinazolinas / Simulação por Computador / Mosquitos Vetores / Inseticidas / Malária / Anopheles Idioma: En Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Arábia Saudita

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Quinazolinas / Simulação por Computador / Mosquitos Vetores / Inseticidas / Malária / Anopheles Idioma: En Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Arábia Saudita