Search details
1.
Diazepinone HBV capsid assembly modulators.
Bioorg Med Chem Lett
; 72: 128823, 2022 09 15.
Article
in English
| MEDLINE | ID: mdl-35644301
2.
Oxadiazepinone HBV capsid assembly modulators.
Bioorg Med Chem Lett
; 52: 128353, 2021 11 15.
Article
in English
| MEDLINE | ID: mdl-34492302
3.
Identification of a new class of HBV capsid assembly modulator.
Bioorg Med Chem Lett
; 39: 127848, 2021 05 01.
Article
in English
| MEDLINE | ID: mdl-33610748
4.
Preclinical Characterization of NVR 3-778, a First-in-Class Capsid Assembly Modulator against Hepatitis B Virus.
Antimicrob Agents Chemother
; 63(1)2019 01.
Article
in English
| MEDLINE | ID: mdl-30373799
5.
SAR studies in the sulfonyl carboxamide class of HBV capsid assembly modulators.
Bioorg Med Chem Lett
; 29(16): 2405-2409, 2019 08 15.
Article
in English
| MEDLINE | ID: mdl-31227344
6.
Hepatitis B Virus Capsid Assembly Modulators, but Not Nucleoside Analogs, Inhibit the Production of Extracellular Pregenomic RNA and Spliced RNA Variants.
Antimicrob Agents Chemother
; 61(8)2017 08.
Article
in English
| MEDLINE | ID: mdl-28559265
7.
Discovery of MK-1832, a Kv1.5 inhibitor with improved selectivity and pharmacokinetics.
Bioorg Med Chem Lett
; 27(4): 1062-1069, 2017 02 15.
Article
in English
| MEDLINE | ID: mdl-28131713
8.
Identification of a methoxynaphthalene scaffold as a core replacement in quinolizidinone amide M(1) positive allosteric modulators.
Bioorg Med Chem Lett
; 24(5): 1417-20, 2014 Mar 01.
Article
in English
| MEDLINE | ID: mdl-24485781
9.
Benzimidazole CB2 agonists: design, synthesis and SAR.
Bioorg Med Chem Lett
; 24(4): 1218-21, 2014 Feb 15.
Article
in English
| MEDLINE | ID: mdl-24461289
10.
Adenosine analogue inhibitors of S-adenosylhomocysteine hydrolase.
Bioorg Med Chem Lett
; 24(12): 2737-40, 2014 Jun 15.
Article
in English
| MEDLINE | ID: mdl-24813734
11.
Discovery of MK-3697: a selective orexin 2 receptor antagonist (2-SORA) for the treatment of insomnia.
Bioorg Med Chem Lett
; 24(20): 4884-90, 2014 Oct 15.
Article
in English
| MEDLINE | ID: mdl-25248679
12.
Discovery of 2,5-diarylnicotinamides as selective orexin-2 receptor antagonists (2-SORAs).
Bioorg Med Chem Lett
; 23(24): 6620-4, 2013 Dec 15.
Article
in English
| MEDLINE | ID: mdl-24215892
13.
Pyridyl aminothiazoles as potent Chk1 inhibitors: optimization of cellular activity.
Bioorg Med Chem Lett
; 22(7): 2613-9, 2012 Apr 01.
Article
in English
| MEDLINE | ID: mdl-22365762
14.
Pyridyl aminothiazoles as potent inhibitors of Chk1 with slow dissociation rates.
Bioorg Med Chem Lett
; 22(7): 2609-12, 2012 Apr 01.
Article
in English
| MEDLINE | ID: mdl-22374217
15.
Discovery of the selective androgen receptor modulator MK-0773 using a rational development strategy based on differential transcriptional requirements for androgenic anabolism versus reproductive physiology.
J Biol Chem
; 285(22): 17054-64, 2010 May 28.
Article
in English
| MEDLINE | ID: mdl-20356837
16.
Quinolizidinone carboxylic acid selective M1 allosteric modulators: SAR in the piperidine series.
Bioorg Med Chem Lett
; 21(6): 1710-5, 2011 Mar 15.
Article
in English
| MEDLINE | ID: mdl-21324684
17.
Fused heterocyclic M1 positive allosteric modulators.
Bioorg Med Chem Lett
; 21(9): 2769-72, 2011 May 01.
Article
in English
| MEDLINE | ID: mdl-21055928
18.
Identification of non-amidine inhibitors of acid-sensing ion channel-3 (ASIC3).
Bioorg Med Chem Lett
; 21(14): 4255-8, 2011 Jul 15.
Article
in English
| MEDLINE | ID: mdl-21669528
19.
High concentration electrophysiology-based fragment screen: discovery of novel acid-sensing ion channel 3 (ASIC3) inhibitors.
Bioorg Med Chem Lett
; 21(9): 2646-9, 2011 May 01.
Article
in English
| MEDLINE | ID: mdl-21257308
20.
Decahydroquinoline amides as highly selective CB2 agonists: role of selectivity on in vivo efficacy in a rodent model of analgesia.
Bioorg Med Chem Lett
; 21(8): 2359-64, 2011 Apr 15.
Article
in English
| MEDLINE | ID: mdl-21420857