1.
J Med Chem
; 50(24): 5882-5, 2007 Nov 29.
Article
in English
| MEDLINE
| ID: mdl-17963373
ABSTRACT
A novel series of antagonists of the human P2X7 receptor is described. Modification of substituents enabled identification of compounds selective for the rat P2X7 receptor and provides useful pharmacological tools for evaluation of the role of P2X7 in disease.