Detalhe da pesquisa
1.
Discovery of a highly potent orally bioavailable imidazo-[1, 2-a]pyrazine Aurora inhibitor.
Bioorg Med Chem Lett
; 28(8): 1397-1403, 2018 05 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29545102
2.
Synthesis and SAR studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off-target kinase selectivity.
Bioorg Med Chem Lett
; 22(10): 3544-9, 2012 May 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22503250
3.
Discovery of novel imidazo[1,2-a]pyrazin-8-amines as Brk/PTK6 inhibitors.
Bioorg Med Chem Lett
; 21(19): 5870-5, 2011 Oct 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21855335
4.
Bioisosteric approach to the discovery of imidazo[1,2-a]pyrazines as potent Aurora kinase inhibitors.
Bioorg Med Chem Lett
; 21(1): 592-8, 2011 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21075632
5.
Discovery of imidazo[1,2-a]pyrazine-based Aurora kinase inhibitors.
Bioorg Med Chem Lett
; 20(17): 5170-4, 2010 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20674350
6.
Discovery of orally bioavailable imidazo[1,2-a]pyrazine-based Aurora kinase inhibitors.
Bioorg Med Chem Lett
; 20(22): 6739-43, 2010 Nov 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20855207
7.
Structure and activity relationships of tartrate-based TACE inhibitors.
Bioorg Med Chem Lett
; 20(16): 4812-5, 2010 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20638281
8.
The discovery of novel tartrate-based TNF-alpha converting enzyme (TACE) inhibitors.
Bioorg Med Chem Lett
; 20(3): 1189-93, 2010 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20022498
9.
Design, Synthesis, and Preclinical Characterization of Selective Factor D Inhibitors Targeting the Alternative Complement Pathway.
J Med Chem
; 62(9): 4656-4668, 2019 05 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-30995036
10.
The Discovery of ( S)-1-(6-(3-((4-(1-(Cyclopropanecarbonyl)piperidin-4-yl)-2-methylphenyl)amino)-2,3-dihydro-1 H-inden-4-yl)pyridin-2-yl)-5-methyl-1 H-pyrazole-4-carboxylic Acid, a Soluble Guanylate Cyclase Activator Specifically Designed for Topical Ocular Delivery as a Therapy for Glaucoma.
J Med Chem
; 61(6): 2552-2570, 2018 03 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-29498522
11.
Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine Core.
ACS Med Chem Lett
; 1(5): 214-8, 2010 Aug 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-24900197
12.
Substrate control of stereoselection in the rhodium(I) catalyzed intramolecular [4 + 2] cycloaddition reaction.
Org Biomol Chem
; 1(12): 2038-40, 2003 Jun 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-12945892