Detalhe da pesquisa
1.
Synthesis of [1-8-NαC]-zanriorb A1, alanine-containing analogues, and their cytotoxic and anti-inflammatory activity.
J Pept Sci
; 28(8): e3405, 2022 Aug.
Artigo
em Inglês
| MEDLINE | ID: mdl-35068012
2.
Synthesis of new clioquinol derivatives as potent α-glucosidase inhibitors; molecular docking, kinetic and structure-activity relationship studies.
Bioorg Chem
; 119: 105506, 2022 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-34896920
3.
Isolation, derivatization, in-vitro, and in-silico studies of potent butyrylcholinesterase inhibitors from Berberis parkeriana Schneid.
Bioorg Chem
; 127: 105944, 2022 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-35905644
4.
Synthesis of 1,2,3,triazole modified analogues of hydrochlorothiazide via click chemistry approach and in-vitro α-glucosidase enzyme inhibition studies.
Mol Divers
; 26(4): 2049-2067, 2022 Aug.
Artigo
em Inglês
| MEDLINE | ID: mdl-34608550
5.
3, 3'- (3, 5-DCPBC) Down-Regulates Multiple Phosphokinase Dependent Signal Transduction Pathways in Malignant Melanoma Cells through Specific Diminution of EGFRY1086 Phosphorylation.
Molecules
; 27(4)2022 Feb 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-35208960
6.
Synthesis of 2-Aminopyrimidine Derivatives and Their Evaluation as ß-Glucuronidase Inhibitors: In Vitro and In Silico Studies.
Molecules
; 27(22)2022 Nov 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-36431887
7.
Dibenzazepine-linked isoxazoles: New and potent class of α-glucosidase inhibitors.
Bioorg Med Chem Lett
; 40: 127979, 2021 05 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-33766763
8.
Distinct genetic landscape and a low response to doxorubicin in a luminal-A breast cancer cell line of Pakistani origin.
Mol Biol Rep
; 48(10): 6821-6829, 2021 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-34495459
9.
On the molecular basis of H2O/DMSO eutectic mixtures by using phenol compounds as molecular sensors: a combined NMR and DFT study.
Phys Chem Chem Phys
; 23(29): 15645-15658, 2021 Aug 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-34268541
10.
Synthesis, crystal structure and Hirshfeld Surface analysis of benzamide derivatives of thiourea as potent inhibitors of α-glucosidase in-vitro.
Bioorg Chem
; 107: 104531, 2021 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-33339666
11.
Identification of new lead molecules against anticancer drug target TFIIH subunit P8 using biophysical and molecular docking studies.
Bioorg Chem
; 114: 105021, 2021 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-34120023
12.
Celebrex derivatives: Synthesis, α-glucosidase inhibition, crystal structures and molecular docking studies.
Bioorg Chem
; 106: 104499, 2021 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-33288319
13.
New isolate from Salvinia molesta with antioxidant and urease inhibitory activity.
Drug Dev Res
; 82(8): 1169-1181, 2021 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-33983647
14.
Stereoselective Synthesis of the Di-Spirooxindole Analogs Based Oxindole and Cyclohexanone Moieties as Potential Anticancer Agents.
Molecules
; 26(20)2021 Oct 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-34684885
15.
Clarithromycin Exerts an Antibiofilm Effect against Salmonella enterica Serovar Typhimurium rdar Biofilm Formation and Transforms the Physiology towards an Apparent Oxygen-Depleted Energy and Carbon Metabolism.
Infect Immun
; 88(11)2020 10 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-32839186
16.
The unique catalytic role of water in aromatic C-H activation at neutral pH: a combined NMR and DFT study of polyphenolic compounds.
Phys Chem Chem Phys
; 22(30): 17401-17411, 2020 Aug 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-32706350
17.
Fungal mediated biotransformation of melengestrol acetate, and T-cell proliferation inhibitory activity of biotransformed compounds.
Bioorg Chem
; 104: 104313, 2020 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-33142425
18.
Insight into the binding affinity of thiourea in the calcium binding pocket of proteinase K, through high resolution X-ray crystallography.
Bioorg Chem
; 94: 103443, 2020 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-31812259
19.
Chemical constituents from Parrotia persica- Structural derivatization and their potential prolyl endopeptidase inhibition activity.
Bioorg Chem
; 96: 103526, 2020 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-32004898
20.
Synthesis and characterisation of thiobarbituric acid enamine derivatives, and evaluation of their α-glucosidase inhibitory and anti-glycation activity.
J Enzyme Inhib Med Chem
; 35(1): 692-701, 2020 Dec.
Artigo
em Inglês
| MEDLINE | ID: mdl-32156165