Detalhe da pesquisa
1.
Direct evaluation of polarity of the ligand binding pocket in retinoid X receptor using a fluorescent solvatochromic agonist.
Bioorg Med Chem Lett
; 96: 129536, 2023 11 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-37913851
2.
Characterization and Interconversion of Two Crystal Forms of NEt-3IB, a Retinoid X Receptor Agonist.
Chem Pharm Bull (Tokyo)
; 71(4): 282-288, 2023.
Artigo
em Inglês
| MEDLINE | ID: mdl-37005253
3.
Fluorescence properties of retinoid X receptor antagonist NEt-SB.
Bioorg Med Chem Lett
; 31: 127666, 2021 01 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-33152377
4.
A partial agonist for retinoid X receptor mitigates experimental colitis.
Int Immunol
; 31(4): 251-262, 2019 03 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-30590577
5.
3H-Imidazo[4,5-b]pyridine-6-carboxylic acid derivatives as rexinoids with reduced teratogenicity.
Bioorg Med Chem Lett
; 29(15): 1891-1894, 2019 08 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-31160175
6.
Fluorine-18 (18F)-labeled retinoidâ¯xâ¯receptor (RXR) partial agonist whose tissue transferability is affected by other RXR ligands.
Bioorg Med Chem
; 27(14): 3128-3134, 2019 07 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31176570
7.
Simple Fluorescence Labeling Method Enables Detection of Intracellular Distribution and Expression Level of Retinoid X Receptors.
ACS Med Chem Lett
; 15(5): 640-645, 2024 May 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-38746897
8.
Structural characterization of 1,3-bis-tert-butyl monocyclic benzene derivatives with agonistic activity towards retinoid X receptor alpha.
Toxicol Lett
; 373: 76-83, 2023 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-36368620
9.
Ligand Screening System for the RXRα Heterodimer Using the Fluorescence RXR Agonist CU-6PMN.
ACS Med Chem Lett
; 14(3): 291-296, 2023 Mar 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-36923911
10.
Increased Molecular Flexibility Widens the Gap between K i and K d values in Screening for Retinoid X Receptor Modulators.
ACS Med Chem Lett
; 13(2): 211-217, 2022 Feb 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-35178177
11.
Identification of a Vitamin-D Receptor Antagonist, MeTC7, which Inhibits the Growth of Xenograft and Transgenic Tumors In Vivo.
J Med Chem
; 65(8): 6039-6055, 2022 04 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-35404047
12.
Creation of Fluorescent RXR Antagonists Based on CBTF-EE and Application to a Fluorescence Polarization Binding Assay.
ACS Med Chem Lett
; 12(6): 1024-1029, 2021 Jun 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-34141088
13.
Discovery of a "Gatekeeper" Antagonist that Blocks Entry Pathway to Retinoid X Receptors (RXRs) without Allosteric Ligand Inhibition in Permissive RXR Heterodimers.
J Med Chem
; 64(1): 430-439, 2021 01 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-33356247
14.
Convenient Retinoid X Receptor Binding Assay Based on Fluorescence Change of the Antagonist NEt-C343.
J Med Chem
; 64(1): 861-870, 2021 01 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-33378197
15.
Competitive Binding Assay with an Umbelliferone-Based Fluorescent Rexinoid for Retinoid X Receptor Ligand Screening.
J Med Chem
; 62(19): 8809-8818, 2019 10 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-31483660
16.
Dual conformation of the ligand induces the partial agonistic activity of retinoid X receptor α (RXRα).
FEBS Lett
; 593(2): 242-250, 2019 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-30565665
17.
Acute lethal toxicity, hyperkalemia associated with renal injury and hepatic damage after intravenous administration of cadmium nitrate in rats.
J Occup Health
; 49(1): 17-24, 2007 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-17314462
18.
Urinary fluoride reference values determined by a fluoride ion selective electrode.
Biol Trace Elem Res
; 119(1): 27-34, 2007 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-17914216
19.
Urinary and serum titanium: assessment as an indicator of exposure to ammonium citratoperoxotitanate (IV) and its influence on renal function.
Biol Trace Elem Res
; 110(2): 119-32, 2006 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-16757841
20.
Urinary yttrium excretion and effects of yttrium chloride on renal function in rats.
Biol Trace Elem Res
; 114(1-3): 225-35, 2006.
Artigo
em Inglês
| MEDLINE | ID: mdl-17206005