Detalhe da pesquisa
1.
Epiminocyclohepta[b]indole analogs as 5-HT6 antagonists.
Bioorg Med Chem Lett
; 22(4): 1494-8, 2012 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22290076
2.
5-(pyridinon-1-yl)indazoles and 5-(furopyridinon-5-yl)indazoles as MCH-1 antagonists.
Bioorg Med Chem Lett
; 20(23): 7015-9, 2010 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20961756
3.
Synthesis and SAR of 4-aryl-1-(indazol-5-yl)pyridin-2(1H)ones as MCH-1 antagonists for the treatment of obesity.
Bioorg Med Chem Lett
; 20(23): 7020-3, 2010 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20951036
4.
Tetrahydrocarboline analogs as MCH-1 antagonists.
Bioorg Med Chem Lett
; 20(23): 7024-8, 2010 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20952195
5.
2,3-Diaminopyrazines as Rho kinase inhibitors.
Bioorg Med Chem Lett
; 20(3): 1137-40, 2010 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20022494
6.
Synthesis and SAR of heterocyclic carboxylic acid isosteres based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesity.
Bioorg Med Chem Lett
; 20(9): 2912-5, 2010 May 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20347296
7.
Discovery of substituted biphenyl imidazoles as potent, bioavailable bombesin receptor subtype-3 agonists.
Bioorg Med Chem Lett
; 20(6): 1913-7, 2010 Mar 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20167483
8.
Synthesis and SAR of derivatives based on 2-biarylethylimidazole as bombesin receptor subtype-3 (BRS-3) agonists for the treatment of obesity.
Bioorg Med Chem Lett
; 20(7): 2074-7, 2010 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20219372
9.
Targeting 5-HT receptors for the treatment of obesity.
Curr Opin Pharmacol
; 11(1): 52-8, 2011 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-21330209
10.
Discovery of MK-5046, a Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Obesity.
ACS Med Chem Lett
; 2(1): 43-7, 2011 Jan 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-24900253