1.
Bioorg Med Chem Lett
; 20(6): 1895-9, 2010 Mar 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-20181479
RESUMO
A series of amide derived beta(3)-adrenergic receptor (AR) agonists is described. The discovery and optimization of several series of compounds derived from 1, is used to lay the SAR foundation for second generation beta(3)-AR agonists for the treatment of overactive bladder.