1.
Bioorg Med Chem Lett
; 14(15): 3869-73, 2004 Aug 02.
Artigo
em Inglês
| MEDLINE
| ID: mdl-15225687
RESUMO
A series of benzoylpyrimidines derived from the anilinepyrimidine CRF(1) antagonists were synthesized. Several synthetic routes were developed to explore the SAR of this series of compounds. Compounds such as 8d (K(i) = 15 nM) exhibited high binding affinities at the human CRF(1) receptor.