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New 2-Ethylthio-4-methylaminoquinazoline derivatives inhibiting two subunits of cytochrome bc1 in Mycobacterium tuberculosis.
Lupien, Andréanne; Foo, Caroline Shi-Yan; Savina, Svetlana; Vocat, Anthony; Piton, Jérémie; Monakhova, Natalia; Benjak, Andrej; Lamprecht, Dirk A; Steyn, Adrie J C; Pethe, Kevin; Makarov, Vadim A; Cole, Stewart T.
Affiliation
  • Lupien A; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Foo CS; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Savina S; Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation.
  • Vocat A; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Piton J; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Monakhova N; Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation.
  • Benjak A; Global Health Institute, Ecole Polytechnique Fédérale de Lausanne, Lausanne, Switzerland.
  • Lamprecht DA; Africa Health Research Institute, Durban, South Africa.
  • Steyn AJC; Africa Health Research Institute, Durban, South Africa.
  • Pethe K; Department of Microbiology, University of Alabama at Birmingham, Birmingham, Alabama, United States of America.
  • Makarov VA; Lee Kong Chian School of Medicine and School of Biological Sciences, Nanyang Technological University, Singapore.
  • Cole ST; Department of Stresses of Microorganisms, A. N. Bach Institute of Biochemistry, Moscow, Russian Federation.
PLoS Pathog ; 16(1): e1008270, 2020 01.
Article in En | MEDLINE | ID: mdl-31971990

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinazolines / Bacterial Proteins / Tuberculosis, Multidrug-Resistant / Electron Transport Complex III / Mycobacterium tuberculosis / Antitubercular Agents Type of study: Prognostic_studies Limits: Humans Language: En Journal: PLoS Pathog Year: 2020 Type: Article Affiliation country: Switzerland

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinazolines / Bacterial Proteins / Tuberculosis, Multidrug-Resistant / Electron Transport Complex III / Mycobacterium tuberculosis / Antitubercular Agents Type of study: Prognostic_studies Limits: Humans Language: En Journal: PLoS Pathog Year: 2020 Type: Article Affiliation country: Switzerland