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Biological evaluation, radiosensitizing activity and structural insights of novel halogenated quinazoline-sulfonamide conjugates as selective human carbonic anhydrases IX/XII inhibitors.
Ghorab, Mostafa M; Soliman, Aiten M; Bua, Silvia; Supuran, Claudiu T.
Affiliation
  • Ghorab MM; Department of Drug Radiation Research, National Center for Radiation Research and Technology (NCRRT), Egyptian Atomic Energy Authority (EAEA), P.O Box 29, Nasr City, Cairo 11765, Egypt. Electronic address: mmsghorab@yahoo.com.
  • Soliman AM; Department of Drug Radiation Research, National Center for Radiation Research and Technology (NCRRT), Egyptian Atomic Energy Authority (EAEA), P.O Box 29, Nasr City, Cairo 11765, Egypt.
  • Bua S; University of Florence, NEUROFARBA Department, Sezione di Scienze Farmaceutiche e Nutraceutiche, Via U. Schiff 6, 50019 Sesto Fiorentino, Florence, Italy.
  • Supuran CT; University of Florence, NEUROFARBA Department, Sezione di Scienze Farmaceutiche e Nutraceutiche, Via U. Schiff 6, 50019 Sesto Fiorentino, Florence, Italy. Electronic address: claudiu.supuran@unifi.it.
Bioorg Chem ; 107: 104618, 2021 02.
Article in En | MEDLINE | ID: mdl-33485104

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinazolines / Radiation-Sensitizing Agents / Carbonic Anhydrase Inhibitors / Carbonic Anhydrases / Carbonic Anhydrase IX Type of study: Prognostic_studies Limits: Humans Language: En Journal: Bioorg Chem Year: 2021 Type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Quinazolines / Radiation-Sensitizing Agents / Carbonic Anhydrase Inhibitors / Carbonic Anhydrases / Carbonic Anhydrase IX Type of study: Prognostic_studies Limits: Humans Language: En Journal: Bioorg Chem Year: 2021 Type: Article