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Structure-Based Design of Potent, Selective, and Orally Bioavailable VPS34 Kinase Inhibitors.
Hu, Dennis X; Patel, Snahel; Chen, Huifen; Wang, Shumei; Staben, Steven T; Dimitrova, Yoana N; Wallweber, Heidi Ackerly; Lee, Joanna Y; Chan, Grace Ka Yan; Sneeringer, Christopher J; Prangley, Madeleine S; Moffat, John G; Wu, Kai C; Schutt, Leah K; Salphati, Laurent; Pang, Jodie; McNamara, Erin; Huang, Haochu; Chen, Yong; Wang, Yunli; Zhao, Wensheng; Lim, Junghyun; Murthy, Aditya; Siu, Michael.
Affiliation
  • Chen Y; Pharmaron Beijing Co., Ltd., 6 Taihe Road, BDA, Beijing 100176, China.
  • Wang Y; Pharmaron Beijing Co., Ltd., 6 Taihe Road, BDA, Beijing 100176, China.
  • Zhao W; Pharmaron Beijing Co., Ltd., 6 Taihe Road, BDA, Beijing 100176, China.
J Med Chem ; 65(17): 11500-11512, 2022 09 08.
Article in En | MEDLINE | ID: mdl-34779204

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Class III Phosphatidylinositol 3-Kinases / Antineoplastic Agents Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2022 Type: Article

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Class III Phosphatidylinositol 3-Kinases / Antineoplastic Agents Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2022 Type: Article