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Novel Labdane Diterpenes-Based Synthetic Derivatives: Identification of a Bifunctional Vasodilator That Inhibits CaV1.2 and Stimulates KCa1.1 Channels.
Carullo, Gabriele; Saponara, Simona; Ahmed, Amer; Gorelli, Beatrice; Mazzotta, Sarah; Trezza, Alfonso; Gianibbi, Beatrice; Campiani, Giuseppe; Fusi, Fabio; Aiello, Francesca.
Affiliation
  • Carullo G; Department of Life Sciences, University of Siena, Via Aldo Moro 2, 53100 Siena, Italy.
  • Saponara S; Department of Life Sciences, University of Siena, Via Aldo Moro 2, 53100 Siena, Italy.
  • Ahmed A; Department of Life Sciences, University of Siena, Via Aldo Moro 2, 53100 Siena, Italy.
  • Gorelli B; Department of Life Sciences, University of Siena, Via Aldo Moro 2, 53100 Siena, Italy.
  • Mazzotta S; Department of Chemistry, University of Milan, Via Golgi 19, 20133 Milano, Italy.
  • Trezza A; Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Via Aldo Moro 2, 53100 Siena, Italy.
  • Gianibbi B; Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Via Aldo Moro 2, 53100 Siena, Italy.
  • Campiani G; Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Via Aldo Moro 2, 53100 Siena, Italy.
  • Fusi F; Department of Biotechnology, Chemistry and Pharmacy, University of Siena, Via Aldo Moro 2, 53100 Siena, Italy.
  • Aiello F; Department of Pharmacy, Health and Nutritional Sciences, University of Calabria, Edif. Polifunzionale, 87036 Arcavacata di Rende, Italy.
Mar Drugs ; 20(8)2022 Aug 13.
Article in En | MEDLINE | ID: mdl-36005518

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Diterpenes / Hypertension Type of study: Diagnostic_studies Limits: Humans Language: En Journal: Mar Drugs Journal subject: BIOLOGIA / FARMACOLOGIA Year: 2022 Type: Article Affiliation country: Italy

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Diterpenes / Hypertension Type of study: Diagnostic_studies Limits: Humans Language: En Journal: Mar Drugs Journal subject: BIOLOGIA / FARMACOLOGIA Year: 2022 Type: Article Affiliation country: Italy