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Small Molecule Degraders of Protein Tyrosine Phosphatase 1B and T-Cell Protein Tyrosine Phosphatase for Cancer Immunotherapy.
Dong, Jiajun; Miao, Jinmin; Miao, Yiming; Qu, Zihan; Zhang, Sheng; Zhu, Peipei; Wiede, Florian; Jassim, Brenson A; Bai, Yunpeng; Nguyen, Quyen; Lin, Jianping; Chen, Lan; Tiganis, Tony; Tao, W Andy; Zhang, Zhong-Yin.
Affiliation
  • Dong J; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University, West Lafayette, IN 47907, USA.
  • Miao J; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University, West Lafayette, IN 47907, USA.
  • Miao Y; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University, West Lafayette, IN 47907, USA.
  • Qu Z; Department of Chemistry, Purdue University, West Lafayette, IN 47907, USA.
  • Zhang S; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University, West Lafayette, IN 47907, USA.
  • Zhu P; Department of Biochemistry, Purdue University, West Lafayette, IN 47907, USA.
  • Wiede F; Monash Biomedicine Discovery Institute, Monash University, Clayton, Victoria, 3800, Australia.
  • Jassim BA; Department of Biochemistry and Molecular Biology, Monash University, Clayton, Victoria, 3800, Australia.
  • Bai Y; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University, West Lafayette, IN 47907, USA.
  • Nguyen Q; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University, West Lafayette, IN 47907, USA.
  • Lin J; Department of Chemistry, Purdue University, West Lafayette, IN 47907, USA.
  • Chen L; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University, West Lafayette, IN 47907, USA.
  • Tiganis T; Institute for Drug Discovery, Purdue University, West Lafayette, IN 47907, USA.
  • Tao WA; Monash Biomedicine Discovery Institute, Monash University, Clayton, Victoria, 3800, Australia.
  • Zhang ZY; Department of Biochemistry and Molecular Biology, Monash University, Clayton, Victoria, 3800, Australia.
Angew Chem Int Ed Engl ; 62(22): e202303818, 2023 05 22.
Article in En | MEDLINE | ID: mdl-36973833

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein Tyrosine Phosphatase, Non-Receptor Type 2 / Neoplasms Limits: Humans Language: En Journal: Angew Chem Int Ed Engl Year: 2023 Type: Article Affiliation country: United States

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Protein Tyrosine Phosphatase, Non-Receptor Type 2 / Neoplasms Limits: Humans Language: En Journal: Angew Chem Int Ed Engl Year: 2023 Type: Article Affiliation country: United States