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Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A.
Leaver, David J; Cleary, Benjamin; Nguyen, Nghi; Priebbenow, Daniel L; Lagiakos, H Rachel; Sanchez, Julie; Xue, Lian; Huang, Fei; Sun, Yuxin; Mujumdar, Prashant; Mudududdla, Ramesh; Varghese, Swapna; Teguh, Silvia; Charman, Susan A; White, Karen L; Katneni, Kasiram; Cuellar, Matthew; Strasser, Jessica M; Dahlin, Jayme L; Walters, Michael A; Street, Ian P; Monahan, Brendon J; Jarman, Kate E; Sabroux, Helene Jousset; Falk, Hendrik; Chung, Matthew C; Hermans, Stefan J; Parker, Michael W; Thomas, Tim; Baell, Jonathan B.
Afiliação
  • Lagiakos HR; Cancer Therapeutics CRC , 343 Royal Parade , Parkville , Victoria 3052 , Australia.
  • Sanchez J; Walter and Eliza Hall Institute of Medical Research , 1G Royal Parade , Parkville , Victoria 3052 , Australia.
  • Xue L; Department of Medical Biology , University of Melbourne , Parkville , Victoria 3050 , Australia.
  • Huang F; School of Pharmaceutical Sciences , Nanjing Tech University , No. 30 South Puzhu Road , Nanjing 211816 , People's Republic of China.
  • Sun Y; School of Pharmaceutical Sciences , Nanjing Tech University , No. 30 South Puzhu Road , Nanjing 211816 , People's Republic of China.
  • Strasser JM; Institute for Therapeutics Discovery and Development , University of Minnesota , 717 Delaware Street SE , Minneapolis , Minnesota 55455 , United States.
  • Dahlin JL; Institute for Therapeutics Discovery and Development , University of Minnesota , 717 Delaware Street SE , Minneapolis , Minnesota 55455 , United States.
  • Walters MA; Department of Pathology , Brigham and Women's Hospital, Boston , 75 Francis Street , Boston , Massachusetts 02115 , United States.
  • Street IP; Institute for Therapeutics Discovery and Development , University of Minnesota , 717 Delaware Street SE , Minneapolis , Minnesota 55455 , United States.
  • Monahan BJ; Walter and Eliza Hall Institute of Medical Research , 1G Royal Parade , Parkville , Victoria 3052 , Australia.
  • Jarman KE; Cancer Therapeutics CRC , 343 Royal Parade , Parkville , Victoria 3052 , Australia.
  • Sabroux HJ; Department of Medical Biology , University of Melbourne , Parkville , Victoria 3050 , Australia.
  • Falk H; Walter and Eliza Hall Institute of Medical Research , 1G Royal Parade , Parkville , Victoria 3052 , Australia.
  • Chung MC; Cancer Therapeutics CRC , 343 Royal Parade , Parkville , Victoria 3052 , Australia.
  • Hermans SJ; Department of Medical Biology , University of Melbourne , Parkville , Victoria 3050 , Australia.
  • Parker MW; Walter and Eliza Hall Institute of Medical Research , 1G Royal Parade , Parkville , Victoria 3052 , Australia.
  • Thomas T; Department of Medical Biology , University of Melbourne , Parkville , Victoria 3050 , Australia.
  • Baell JB; Walter and Eliza Hall Institute of Medical Research , 1G Royal Parade , Parkville , Victoria 3052 , Australia.
J Med Chem ; 62(15): 7146-7159, 2019 08 08.
Article em En | MEDLINE | ID: mdl-31256587

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzenossulfonatos / Histona Acetiltransferases / Descoberta de Drogas / Hidrazinas Limite: Animals / Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzenossulfonatos / Histona Acetiltransferases / Descoberta de Drogas / Hidrazinas Limite: Animals / Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2019 Tipo de documento: Article