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Optimization of 5-substituted thiazolyl ureas and 6-substituted imidazopyridines as potential HIV-1 latency reversing agents.
Nguyen, William; Jacobson, Jonathan; Jarman, Kate E; Blackmore, Timothy R; Sabroux, Helene Jousset; Lewin, Sharon R; Purcell, Damian F; Sleebs, Brad E.
Afiliação
  • Nguyen W; The Walter and Eliza Hall Institute for Medical Research, Parkville, Victoria, 3052, Australia; Department of Medical Biology, University of Melbourne, Parkville, Victoria, 3052, Australia.
  • Jacobson J; Department of Microbiology and Immunology, University of Melbourne at the Peter Doherty Institute of Infection and Immunity, University of Melbourne, Parkville, Victoria, 3000, Australia.
  • Jarman KE; The Walter and Eliza Hall Institute for Medical Research, Parkville, Victoria, 3052, Australia; Department of Medical Biology, University of Melbourne, Parkville, Victoria, 3052, Australia.
  • Blackmore TR; The Walter and Eliza Hall Institute for Medical Research, Parkville, Victoria, 3052, Australia; Department of Medical Biology, University of Melbourne, Parkville, Victoria, 3052, Australia.
  • Sabroux HJ; The Walter and Eliza Hall Institute for Medical Research, Parkville, Victoria, 3052, Australia; Department of Medical Biology, University of Melbourne, Parkville, Victoria, 3052, Australia.
  • Lewin SR; Department of Microbiology and Immunology, University of Melbourne at the Peter Doherty Institute of Infection and Immunity, University of Melbourne, Parkville, Victoria, 3000, Australia; The Peter Doherty Institute for Infection and Immunity, The University of Melbourne and Royal Melbourne Hospital
  • Purcell DF; Department of Microbiology and Immunology, University of Melbourne at the Peter Doherty Institute of Infection and Immunity, University of Melbourne, Parkville, Victoria, 3000, Australia.
  • Sleebs BE; The Walter and Eliza Hall Institute for Medical Research, Parkville, Victoria, 3052, Australia; Department of Medical Biology, University of Melbourne, Parkville, Victoria, 3052, Australia. Electronic address: sleebs@wehi.edu.au.
Eur J Med Chem ; 195: 112254, 2020 Jun 01.
Article em En | MEDLINE | ID: mdl-32251744

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piridinas / Tiazóis / Ureia / HIV-1 / Latência Viral / Imidazóis Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Austrália

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piridinas / Tiazóis / Ureia / HIV-1 / Latência Viral / Imidazóis Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Austrália