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Discovery of Selective Small-Molecule Inhibitors for the ENL YEATS Domain.
Ma, Xinyu R; Xu, Longxia; Xu, Shiqing; Klein, Brianna J; Wang, Hongkuan; Das, Sukant; Li, Kuai; Yang, Kai S; Sohail, Sana; Chapman, Andrew; Kutateladze, Tatiana G; Shi, Xiaobing; Liu, Wenshe Ray; Wen, Hong.
Afiliação
  • Ma XR; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, Texas 77843, United States.
  • Xu L; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, United States.
  • Xu S; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, Texas 77843, United States.
  • Klein BJ; Department of Pharmacology, University of Colorado School of Medicine, Aurora, Colorado 80045, United States.
  • Wang H; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, United States.
  • Das S; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, Texas 77843, United States.
  • Li K; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, United States.
  • Yang KS; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, Texas 77843, United States.
  • Sohail S; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, United States.
  • Chapman A; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, Texas 77843, United States.
  • Kutateladze TG; Department of Pharmacology, University of Colorado School of Medicine, Aurora, Colorado 80045, United States.
  • Shi X; Department of Epigenetics, Van Andel Institute, Grand Rapids, Michigan 49503, United States.
  • Liu WR; Texas A&M Drug Discovery Laboratory, Department of Chemistry, Texas A&M University, College Station, Texas 77843, United States.
  • Wen H; Institute of Biosciences and Technology and Department of Translational Medical Sciences, College of Medicine, Texas A&M University, Houston, Texas 77030, United States.
J Med Chem ; 64(15): 10997-11013, 2021 08 12.
Article em En | MEDLINE | ID: mdl-34279931

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leucemia Mieloide Aguda / Fatores de Elongação da Transcrição / Bibliotecas de Moléculas Pequenas / Descoberta de Drogas / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leucemia Mieloide Aguda / Fatores de Elongação da Transcrição / Bibliotecas de Moléculas Pequenas / Descoberta de Drogas / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Estados Unidos