Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1.

Hall, Adrian; Abendroth, Jan; Bolejack, Madison J; Ceska, Tom; Dell'Aiera, Sylvie; Ellis, Victoria; Fox, David; François, Cyril; Muruthi, Muigai M; Prével, Camille; Poullennec, Karine; Romanov, Sergei; Valade, Anne; Vanbellinghen, Alain; Yano, Jason; Geraerts, Martine

Hall, Adrian; Abendroth, Jan; Bolejack, Madison J; Ceska, Tom; Dell'Aiera, Sylvie; Ellis, Victoria; Fox, David; François, Cyril; Muruthi, Muigai M; Prével, Camille; Poullennec, Karine; Romanov, Sergei; Valade, Anne; Vanbellinghen, Alain; Yano, Jason; Geraerts, Martine.

Afiliação

Hall A; UCB, Avenue de l'Industrie, Braine-L'Alleud 1420, Belgium.
Abendroth J; UCB Seattle, 7869 NE Day Road West, Bainbridge Island, Washington 98110, United States.
Bolejack MJ; UCB Seattle, 7869 NE Day Road West, Bainbridge Island, Washington 98110, United States.
Ceska T; UCB, 216 Bath Road, Slough SL1 3WE, U.K.
Dell'Aiera S; UCB, Avenue de l'Industrie, Braine-L'Alleud 1420, Belgium.
Ellis V; UCB, 216 Bath Road, Slough SL1 3WE, U.K.
Fox D; UCB Seattle, 7869 NE Day Road West, Bainbridge Island, Washington 98110, United States.
François C; NovAliX, Avenue de l'Industrie, Braine-L'Alleud 1420, Belgium.
Muruthi MM; UCB Seattle, 7869 NE Day Road West, Bainbridge Island, Washington 98110, United States.
Prével C; UCB, Avenue de l'Industrie, Braine-L'Alleud 1420, Belgium.
Poullennec K; UCB, Avenue de l'Industrie, Braine-L'Alleud 1420, Belgium.
Romanov S; NANOSYN, 3100 Central Expressway, Santa Clara, California 95051, United States.
Valade A; UCB, Avenue de l'Industrie, Braine-L'Alleud 1420, Belgium.
Vanbellinghen A; UCB, Avenue de l'Industrie, Braine-L'Alleud 1420, Belgium.
Yano J; UCB Boston, 87 Cambridge Park Drive, Cambridge, Massachusetts 02140, United States.
Geraerts M; UCB, Avenue de l'Industrie, Braine-L'Alleud 1420, Belgium.

ACS Med Chem Lett ; 13(7): 1099-1108, 2022 Jul 14.

Article em En | MEDLINE | ID: mdl-35859861

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Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Bélgica

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