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Synthesis and structure-activity relationship of new nicotinamide phosphoribosyltransferase inhibitors with antitumor activity on solid and haematological cancer.
Fratta, Simone; Biniecka, Paulina; Moreno-Vargas, Antonio J; Carmona, Ana T; Nahimana, Aimable; Duchosal, Michel A; Piacente, Francesco; Bruzzone, Santina; Caffa, Irene; Nencioni, Alessio; Robina, Inmaculada.
Afiliação
  • Fratta S; Departamento de Química Orgánica, Facultad de Química, Universidad de Sevilla, Sevilla, 41012, Spain.
  • Biniecka P; Central Laboratory of Hematology, Medical Laboratory and Pathology Department, Lausanne University Hospital, 1011, Lausanne, Switzerland.
  • Moreno-Vargas AJ; Departamento de Química Orgánica, Facultad de Química, Universidad de Sevilla, Sevilla, 41012, Spain.
  • Carmona AT; Departamento de Química Orgánica, Facultad de Química, Universidad de Sevilla, Sevilla, 41012, Spain. Electronic address: anatere@us.es.
  • Nahimana A; Central Laboratory of Hematology, Medical Laboratory and Pathology Department, Lausanne University Hospital, 1011, Lausanne, Switzerland.
  • Duchosal MA; Central Laboratory of Hematology, Medical Laboratory and Pathology Department, Lausanne University Hospital, 1011, Lausanne, Switzerland; Service of Hematology, Oncology Department, Lausanne University Hospital, 1011, Lausanne, Switzerland.
  • Piacente F; Department of Experimental Medicine, Section of Biochemistry, University of Genoa, 16132, Genoa, Italy.
  • Bruzzone S; Department of Experimental Medicine, Section of Biochemistry, University of Genoa, 16132, Genoa, Italy.
  • Caffa I; Department of Internal Medicine and Medical Specialties, University of Genoa, 16132, Genoa, Italy; IRCCS Ospedale Policlinico San Martino, 16132, Genoa, Italy.
  • Nencioni A; Department of Internal Medicine and Medical Specialties, University of Genoa, 16132, Genoa, Italy; IRCCS Ospedale Policlinico San Martino, 16132, Genoa, Italy.
  • Robina I; Departamento de Química Orgánica, Facultad de Química, Universidad de Sevilla, Sevilla, 41012, Spain. Electronic address: robina@us.es.
Eur J Med Chem ; 250: 115170, 2023 Mar 15.
Article em En | MEDLINE | ID: mdl-36787658

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leucemia / Neoplasias Hematológicas / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Espanha

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leucemia / Neoplasias Hematológicas / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Espanha