1.
Chem Commun (Camb)
; 55(9): 1310-1313, 2019 Jan 24.
Artículo
en Inglés
| MEDLINE
| ID: mdl-30633279
RESUMEN
The first application of sulfo-click chemistry with 18F-labeled thio acids is described. The simple one-pot/three-component reaction proceeded rapidly within 30 min using mild reaction conditions to give various 18F-labeled small molecule N-acylsulfonamides in radiochemical conversions of 38-99%, and radiolabeled peptides in 20-25% isolated and decay-corrected radiochemical yields.