1.
Org Lett
; 26(19): 4043-4048, 2024 May 17.
Article
in English
| MEDLINE
| ID: mdl-38695368
ABSTRACT
A radical ring-opening arylation of cyclopropanol with 1,2,3-triazole has been achieved. This synthetic protocol provides straightforward access to a wide range of structurally diverse and chiral 4,5,6,7-tetrahydro[1,2,3]triazolo[1,5-a]pyridines with high efficiency from readily available chiral cyclopropanols.