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Molecules ; 26(21)2021 Oct 21.
Article in English | MEDLINE | ID: mdl-34770776

ABSTRACT

PDZ (postsynaptic density (PSD95), discs large (Dlg), and zonula occludens (ZO-1)-dependent interactions are widely distributed within different cell types and regulate a variety of cellular processes. To date, some of these interactions have been identified as targets of small molecules or peptides, mainly related to central nervous system disorders and cancer. Recently, the knowledge of PDZ proteins and their interactions has been extended to various cell types of the immune system, suggesting that their targeting by viral pathogens may constitute an immune evasion mechanism that favors viral replication and dissemination. Thus, the pharmacological modulation of these interactions, either with small molecules or peptides, could help in the control of some immune-related diseases. Deeper structural and functional knowledge of this kind of protein-protein interactions, especially in immune cells, will uncover novel pharmacological targets for a diversity of clinical conditions.


Subject(s)
PDZ Domains/drug effects , Peptides/chemistry , Peptides/pharmacology , Protein Interaction Domains and Motifs/drug effects , Animals , Disease Management , Disease Susceptibility , Humans , Immune System Diseases/drug therapy , Immune System Diseases/etiology , Immune System Diseases/metabolism , Models, Molecular , Molecular Targeted Therapy , Peptides/therapeutic use , Protein Binding/drug effects , Protein Conformation , Structure-Activity Relationship
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