1.
Bioorg Med Chem Lett
; 18(20): 5428-30, 2008 Oct 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-18818075
RESUMEN
A series of pyrazolo[1,5-a]pyridine derivatives was designed and synthesized as novel potent p38 kinase inhibitors. Our approaches towards improving in vitro metabolism and in vivo pharmacokinetic properties of the series are described.