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Bioorg Med Chem Lett
; 12(1): 65-8, 2002 Jan 07.
Artículo
en Inglés
| MEDLINE
| ID: mdl-11738574
RESUMEN
A series of 4-aryl/cycloalkyl-5-phenyloxazole derivatives was synthesized and evaluated for their ability to inhibit cyclooxygenase-2 (COX-2) and cyclooxygenase-1 (COX-1). These compounds were found to be potent and selective COX-2 inhibitors.